| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA700689 | F | Percent of compound radioactivity ([3H]-Ap4A Degradation), determined in the incubation medium of INS-1 cell membranes | 5 | ALA1144917 | cell-based format | Scientific Literature | ||
| 2. | ALA700690 | F | Percent of compound radioactivity ([3H]-Ap4A Degradation), in presence of added Ap(s)pCH2pp(s)A, in the incubation medium of INS-1 cell membranes | 4 | ALA1144917 | cell-based format | Scientific Literature | ||
| 3. | ALA700691 | F | Percent of compound radioactivity ([3H]-Ap4A Degradation), in presence of added Ap(s)pCHClpp(s)A, in the incubation medium of INS-1 cell membranes | 3 | ALA1144917 | cell-based format | Scientific Literature | ||
| 4. | ALA700692 | F | Percent of compound radioactivity ([3H]-Ap4A Degradation), in presence of added Ap4A, in the incubation medium of INS-1 cell membranes | 5 | ALA1144917 | cell-based format | Scientific Literature | ||
| 5. | ALA751806 | F | Antagonist activity against recombinant human P2X purinoceptor 3 (P2X3 ) | 11 | ALA1135773 | assay format | Scientific Literature | ||
| 6. | ALA750982 | F | Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4) | 8 | ALA1135773 | assay format | Scientific Literature | ||
| 7. | ALA751765 | F | Evaluated for agonist activity against phospholipase C coupled recombinant human P2Y purinoceptor 2 (P2Y2) | 12 | ALA1135773 | assay format | Scientific Literature | ||
| 8. | ALA757043 | F | The compound was evaluated for antagonist activity against phospholipase C coupled recombinant rat P2Y purinoceptor 4 (P2Y4) | 2 | ALA1135773 | assay format | Scientific Literature | ||
| 9. | ALA759509 | F | Antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 ) | 11 | ALA1135773 | assay format | Scientific Literature | ||
| 10. | ALA759522 | F | The compound was evaluated for antagonist activity against recombinant human receptor P2X purinoceptor 2 (P2X2 ) | 3 | ALA1135773 | assay format | Scientific Literature | ||
| 11. | ALA798157 | F | Percent of compound radioactivity ([3H]-Ap4A Degradation) in heparinized rat plasma (saline) | Rattus norvegicus | 5 | ALA1144917 | organism-based format | Scientific Literature | |
| 12. | ALA798158 | F | Percent of compound radioactivity ([3H]-Ap4A Degradation), in presence of added Ap(s)pCH2pp(s)A, in heparinized rat plasma | Rattus norvegicus | 5 | ALA1144917 | organism-based format | Scientific Literature | |
| 13. | ALA878010 | F | Percent of compound radioactivity ([3H]-Ap4A Degradation), in presence of added Ap(s)pCHClpp(s)A, in heparinized rat plasma | Rattus norvegicus | 5 | ALA1144917 | organism-based format | Scientific Literature | |
| 14. | ALA971528 | B | Ratio of EC50 for N-terminal HA epitope-tagged human P2Y2 receptor C278S mutant to EC50 for wild type 3 human P2Y2 receptor | Homo sapiens | 4 | ALA1138525 | single protein format | Scientific Literature | |
| 15. | ALA971531 | F | Agonist activity at N-terminal HA epitope-tagged human P2Y2 receptor C278S mutant expressed in human 1321N1 cells assessed as increase in intracellular calcium level | Homo sapiens | 4 | ALA1138525 | cell-based format | Scientific Literature | |
| 16. | ALA971534 | F | Agonist activity at N-terminal HA epitope-tagged human P2Y2 receptor S296A mutant expressed in human 1321N1 cells assessed as increase in intracellular calcium level relative to carbachol | Homo sapiens | 4 | ALA1138525 | cell-based format | Scientific Literature | |
| 17. | ALA971535 | F | Agonist activity at N-terminal HA epitope-tagged human P2Y2 receptor S296A mutant expressed in human 1321N1 cells assessed as increase in intracellular calcium level | Homo sapiens | 4 | ALA1138525 | cell-based format | Scientific Literature | |
| 18. | ALA971536 | F | Agonist activity at N-terminal HA epitope-tagged wild type 3 human P2Y2 receptor expressed in human 1321N1 cells assessed as increase in intracellular calcium level relative to carbachol | Homo sapiens | 4 | ALA1138525 | cell-based format | Scientific Literature | |
| 19. | ALA971541 | F | Agonist activity at N-terminal HA epitope-tagged wild type 3 human P2Y2 receptor expressed in human 1321N1 cells assessed as increase in intracellular calcium level | Homo sapiens | 5 | ALA1138525 | cell-based format | Scientific Literature | |
| 20. | ALA974435 | F | Agonist activity at N-terminal HA epitope-tagged wild type 4 human P2Y2 receptor expressed in human 1321N1 cells assessed as increase in intracellular calcium level | Homo sapiens | 4 | ALA1138525 | cell-based format | Scientific Literature |
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