| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3868326 | ADME | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 21 | ALA3867477 | single protein format | Scientific Literature | |
| 2. | ALA3868329 | Binding | Inhibition of Cav1.2 (unknown origin) | Homo sapiens | 24 | ALA3867477 | single protein format | Scientific Literature | |
| 3. | ALA3868334 | ADME | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 21 | ALA3867477 | single protein format | Scientific Literature | |
| 4. | ALA3868338 | Binding | Displacement of (2S)-N-(2-phenylphenyl)-1-[2-[1-(tritritiomethyl)benzimidazol-2-yl]sulfanylacetyl]pyrrolidine-2-carboxamide from human OX1 receptor Ile408-Val mutant expressed on CHO cell membrane measured after 3 hrs by TopCount method | Homo sapiens | 48 | ALA3867477 | cell-based format | Scientific Literature | |
| 5. | ALA3868339 | Binding | Displacement of (2S)-N-(2-pyrrol-1-ylphenyl)-1-[2-[1-(tritritiomethyl)benzimidazol-2-yl]sulfanylacetyl]pyrrolidine-2-carboxamide from human OX2 receptor expressed on CHO cell membrane measured after 3 hrs by TopCount method | Homo sapiens | 48 | ALA3867477 | cell-based format | Scientific Literature | |
| 6. | ALA3868340 | Binding | Selectivity index, ratio of Ki for human OX2 receptor expressed on CHO cell membrane to Ki for Ile408-Val variant human OX1 receptor expressed on CHO cell membrane | Homo sapiens | 46 | ALA3867477 | cell-based format | Scientific Literature | |
| 7. | ALA3868375 | Physicochemical | Solubility of the compound | 22 | ALA3867477 | small-molecule physicochemical format | Scientific Literature |
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