| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3860801 | Functional | Agonist activity at human KISS1R expressed in CHO/dhfr cells assessed as increase in intracellular Ca2+ levels measured for 180 secs by Fluo 3-AM dye based FLIPR assay | Homo sapiens | 36 | ALA3860048 | cell-based format | Scientific Literature | |
| 2. | ALA3860802 | Functional | Agonist activity at rat KISS1R expressed in CHO/dhfr cells assessed as increase in intracellular Ca2+ levels measured for 180 secs by Fluo 3-AM dye based FLIPR assay | Rattus norvegicus | 36 | ALA3860048 | cell-based format | Scientific Literature | |
| 3. | ALA3860803 | Functional | Inhibition of testosterone levels in CD(SD) rat assessed as plasma testosterone level <0.04 ng/ml at 0.1 nmol/hr, sc administered continuously for 6 days through alzet osmotic pump measured after 6 days by radio-immunoassay | Rattus norvegicus | 35 | ALA3860048 | organism-based format | Scientific Literature | |
| 4. | ALA3860804 | Functional | Inhibition of testosterone levels in CD(SD) rat assessed as plasma testosterone level <0.04 ng/ml at 0.03 nmol/hr, sc administered continuously for 6 days through alzet osmotic pump measured after 6 days by radio-immunoassay | Rattus norvegicus | 30 | ALA3860048 | organism-based format | Scientific Literature | |
| 5. | ALA3860805 | Functional | Inhibition of testosterone levels in CD(SD) rat assessed as plasma testosterone level <0.04 ng/ml at 0.01 nmol/hr, sc administered continuously for 6 days through alzet osmotic pump measured after 6 days by radio-immunoassay | Rattus norvegicus | 28 | ALA3860048 | organism-based format | Scientific Literature | |
| 6. | ALA3860806 | Functional | Inhibition of testosterone levels in CD(SD) rat assessed as plasma testosterone level <0.04 ng/ml at 0.003 nmol/hr, sc administered continuously for 6 days through alzet osmotic pump measured after 6 days by radio-immunoassay | Rattus norvegicus | 35 | ALA3860048 | organism-based format | Scientific Literature | |
| 7. | ALA3860823 | Physicochemical | Solubility of the compound in water at 20 mg/ml | 7 | ALA3860048 | small-molecule physicochemical format | Scientific Literature |
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