# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3883065 | Binding | Inhibition of recombinant human N-terminal His6-tagged EphA2 (N598 to R890 residues) expressed in baculovirus using poly-EY as substrate after 180 mins by luciferase coupled chemiluminescence assay | Homo sapiens | 325 | ALA3882729 | assay format | Patent Bioactivity Data | |
2. | ALA3883066 | Binding | Inhibition of recombinant human N-terminal His6-tagged EphB4 kinase domain (E605 to E890 residues) expressed in baculovirus using poly-AEKY as substrate after 150 mins in presence of gamma33P-ATP by liquid scintillation spectrometry | Homo sapiens | 344 | ALA3882729 | assay format | Patent Bioactivity Data | |
3. | ALA3883067 | Binding | Inhibition of recombinant human N-terminal GST His6-tagged thrombin cleavage site-fused EGFR (H672 to A1210 residues) expressed in baculovirus using poly-EY as substrate after 210 mins by luciferase coupled chemiluminescence assay | Homo sapiens | 327 | ALA3882729 | assay format | Patent Bioactivity Data | |
4. | ALA3883068 | Binding | Inhibition of recombinant human N-terminal GST His6-tagged thrombin cleavage site-fused ErbB2 kinase domain (Q679 to V1255 residues) expressed in baculovirus infected insect Sf9 cells using biotinylated poly-EY as substrate after 60 mins by alphascreen assay | Homo sapiens | 157 | ALA3882729 | cell-based format | Patent Bioactivity Data | |
5. | ALA3883069 | Binding | Inhibition of recombinant human N-terminal GST-fused KDR (D807 to V1356 residues) expressed in baculovirus infected Escherichia coli or insect Sf9 cells using poly-EY as substrate after 240 mins by luciferase coupled chemiluminescence assay | Homo sapiens | 327 | ALA3882729 | cell-based format | Patent Bioactivity Data | |
6. | ALA3883070 | Binding | Inhibition of recombinant human N-terminal GST-tagged factor 10a cleavage site-fused Flt1 (K784 to I1338 residues) expressed in baculovirus infected insect Sf9 cells using poly-EY as substrate after 120 mins in presence of gamma33P-ATP by liquid scintillation spectrometry | Homo sapiens | 55 | ALA3882729 | cell-based format | Patent Bioactivity Data |