# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4035836 | B | Inhibition of recombinant human N-terminal FLAG-tagged KDM5A expressed in baculovirus infected Sf9 insect cells using H3K4me3 peptide as substrate after 30 to 45 mins by TR-FRET assay | Homo sapiens | 39 | ALA4033700 | cell-based format | Scientific Literature | |
2. | ALA4035843 | B | Inhibition of KDM5A in human PC9 cells assessed as increase in H3K4me3 level after 5 days by mass-spectrometric method | Homo sapiens | 9 | ALA4033700 | cell-based format | Scientific Literature | |
3. | ALA5237427 | B | Inhibition of KDM5A (unknown origin ) by Alphascreen assay | Homo sapiens | 16 | ALA5236557 | single protein format | Scientific Literature | |
4. | ALA5237433 | F | Antiproliferative activity against human PC-9 cells assessed as reduction in cell viability | Homo sapiens | 7 | ALA5236557 | cell-based format | Scientific Literature |