| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4054226 | B | Inhibition of full-length mouse 11beta-HSD1 expressed in HEK293 microsomal fraction using [3H]cortisone as substrate after 1 hr by scintillation proximity assay | Mus musculus | 7 | ALA4052631 | assay format | Scientific Literature | |
| 2. | ALA4054227 | B | Inhibition of full-length mouse 11beta-HSD1 expressed in HEK293 microsomal fraction at 1 uM using [3H]cortisone as substrate after 1 hr by scintillation proximity assay relative to control | Mus musculus | 36 | ALA4052631 | assay format | Scientific Literature | |
| 3. | ALA4054228 | B | Inhibition of full-length human 11beta-HSD1 expressed in HEK293 microsomal fraction at 1 uM using [3H]cortisone as substrate after 2 hr by scintillation proximity assay relative to control | Homo sapiens | 36 | ALA4052631 | cell-based format | Scientific Literature | |
| 4. | ALA4054230 | B | Inhibition of full-length mouse 11beta-HSD2 expressed in HEK293 microsomal fraction using [3H]cortisone as substrate after 1 hr by scintillation proximity assay | Mus musculus | 6 | ALA4052631 | assay format | Scientific Literature | |
| 5. | ALA4054233 | B | Selectivity index, ratio of IC50 for mouse full length 11beta-HSD2 expressed in HEK293 microsomal fraction to IC50 for mouse full length 11beta-HSD1 expressed in HEK293 microsomal fraction | Mus musculus | 6 | ALA4052631 | assay format | Scientific Literature |
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