| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4023943 | P | Dissociation constant, pKa of the compound by capillary electrophoresis | 14 | small-molecule physicochemical format | Scientific Literature | |||
| 2. | ALA4023962 | B | Allosteric activation of human AMPK alpha1/beta1/gamma1 by TR-FRET assay | Homo sapiens | 14 | protein complex format | Scientific Literature | ||
| 3. | ALA4023963 | B | Allosteric activation of human AMPK alpha1/beta1/gamma1 by TR-FRET assay relative to maximum activation of AMP | Homo sapiens | 14 | protein complex format | Scientific Literature | ||
| 4. | ALA4023964 | B | Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assay | Homo sapiens | 14 | protein complex format | Scientific Literature | ||
| 5. | ALA4023965 | P | Lipophilicity, log D of compound at pH 7.4 by shake-flask method | 14 | small-molecule physicochemical format | Scientific Literature | |||
| 6. | ALA4023966 | A | Apparent permeability from apical to basolateral in RRCK cells after 1 hr by LC-MS analysis | Canis lupus familiaris | 14 | cell-based format | Scientific Literature | ||
| 7. | ALA4023967 | A | Total intrinsic clearance in human hepatocytes assessed as per million cells at 1 uM after 4 hrs by LC-MS/MS analysis | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 8. | ALA4023968 | A | Substrate activity at human OAT3 expressed in HEK293 cells assessed as ratio of compound uptake in human OAT3 transfected HEK293 cells to uptake in vector-treated HEK293 cells at 1 uM after 3 mins by LC-MS analysis | Homo sapiens | 14 | cell-based format | Scientific Literature |
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