# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4031690 | B | Inhibition of human GAT3 L314Q mutant expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
2. | ALA4031691 | P | Solubility of compound in pH 7.4 phosphate buffer after 24 hrs by HPLC-UV method | 6 | small-molecule physicochemical format | Scientific Literature | |||
3. | ALA4031696 | B | Inhibition of human GAT1 expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 36 | cell-based format | Scientific Literature | ||
4. | ALA4031697 | B | Inhibition of human BGT1 expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 33 | cell-based format | Scientific Literature | ||
5. | ALA4031698 | B | Inhibition of human GAT2 expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 32 | cell-based format | Scientific Literature | ||
6. | ALA4031699 | B | Inhibition of human GAT3 expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 32 | cell-based format | Scientific Literature | ||
7. | ALA4031700 | B | Inhibition of mouse GAT1 expressed in HEK293 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Mus musculus | 39 | cell-based format | Scientific Literature | ||
8. | ALA4031701 | B | Inhibition of mouse BGT1 expressed in HEK293 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Mus musculus | 42 | cell-based format | Scientific Literature | ||
9. | ALA4031702 | B | Inhibition of mouse GAT2 expressed in HEK293 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Mus musculus | 42 | cell-based format | Scientific Literature | ||
10. | ALA4031703 | B | Inhibition of mouse GAT3 expressed in HEK293 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Mus musculus | 42 | cell-based format | Scientific Literature | ||
11. | ALA4031705 | B | Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cell membranes at 10 uM after 90 mins by scintillation counting method | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
12. | ALA4031706 | B | Displacement of [3H]SCH23390 from human Dopamine receptor D1 receptor expressed in HEKT cell membranes at 10 uM after 90 mins by scintillation counting method | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
13. | ALA4031707 | B | Displacement of [3H]N-methylspiperone from human Dopamine receptor D2 receptor expressed in fibroblast cell membranes at 10 uM after 90 mins by scintillation counting method | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
14. | ALA4031708 | B | Displacement of [3H]N-methylspiperone from human Dopamine receptor D4 receptor at 10 uM after 90 mins by scintillation counting method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
15. | ALA4031711 | B | Binding affinity to sigma receptor (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
16. | ALA4031712 | B | Inhibition of human BGT1 F295Y mutant expressed in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
17. | ALA4031713 | B | Inhibition of human BGT1 Q299L mutant expressed in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
18. | ALA4031714 | B | Inhibition of human BGT1 K310N mutant expressed in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
19. | ALA4031715 | B | Inhibition of human BGT1 H312N mutant expressed in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
20. | ALA4031716 | B | Inhibition of human BGT1 K317R mutant expressed in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 3 | cell-based format | Scientific Literature |