| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4036811 | B | Activation of KCNQ2/3 (unknown origin) | Homo sapiens | 3 | ALA4033760 | protein complex format | Scientific Literature | |
| 2. | ALA4036812 | B | Inhibition of KCNQ1 (unknown origin) | Homo sapiens | 3 | ALA4033760 | single protein format | Scientific Literature | |
| 3. | ALA4036813 | B | Inhibition of full length human TRPA1 at a holding potential of 15 mV measured after 1 min by PatchXpress electrophysiology assay | Homo sapiens | 27 | ALA4033760 | single protein format | Scientific Literature | |
| 4. | ALA4036814 | B | Inhibition of full length opossum TRPA1 at a holding potential of 15 mV measured after 1 min by PatchXpress electrophysiology assay | Monodelphis domestica | 1 | ALA4033760 | assay format | Scientific Literature | |
| 5. | ALA4036815 | B | Inhibition of full length rat TRPA1 at a holding potential of 15 mV measured after 1 min by PatchXpress electrophysiology assay | Rattus norvegicus | 27 | ALA4033760 | single protein format | Scientific Literature | |
| 6. | ALA4036816 | B | Inhibition of full length opossum TRPA1 hS5 chimera at a holding potential of 15 mV measured after 1 min by PatchXpress electrophysiology assay | Monodelphis domestica | 1 | ALA4033760 | assay format | Scientific Literature | |
| 7. | ALA4036817 | B | Inhibition of full length human TRPA1 oS5 chimera at a holding potential of 15 mV measured after 1 min by PatchXpress electrophysiology assay | Homo sapiens | 1 | ALA4033760 | single protein format | Scientific Literature | |
| 8. | ALA4036818 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 2 | ALA4033760 | assay format | Scientific Literature | |
| 9. | ALA4036819 | A | Intrinsic clearance in rat liver microsomes | Rattus norvegicus | 2 | ALA4033760 | assay format | Scientific Literature | |
| 10. | ALA4036820 | A | Permeability across basolateral to apical side in RRCK cells expressing MDR1 | Canis lupus familiaris | 2 | ALA4033760 | cell-based format | Scientific Literature | |
| 11. | ALA4036821 | A | Permeability across apical to basolateral side in RRCK cells expressing MDR1 | Canis lupus familiaris | 2 | ALA4033760 | cell-based format | Scientific Literature | |
| 12. | ALA4036822 | A | Efflux ratio of permeability from apical to basolateral over basolateral to apical in RRCK cells expressing MDR1 | Canis lupus familiaris | 2 | ALA4033760 | cell-based format | Scientific Literature | |
| 13. | ALA4036823 | P | Aqueous solubility of the compound by kinetic miniaturized shakeflask method | 2 | ALA4033760 | small-molecule physicochemical format | Scientific Literature | ||
| 14. | ALA4036824 | B | Antagonist activity at human TRPA1 by calcium flux based FLIPR assay | Homo sapiens | 3 | ALA4033760 | single protein format | Scientific Literature | |
| 15. | ALA4036825 | B | Inhibition of human ERG | Homo sapiens | 3 | ALA4033760 | single protein format | Scientific Literature | |
| 16. | ALA4036826 | B | Inhibition of Nav1.5 (unknown origin) | Homo sapiens | 3 | ALA4033760 | single protein format | Scientific Literature | |
| 17. | ALA4036827 | B | Inhibition of Nav1.7 (unknown origin) | Homo sapiens | 2 | ALA4033760 | single protein format | Scientific Literature | |
| 18. | ALA4036828 | B | Inhibition of TRPV1 (unknown origin) | Homo sapiens | 3 | ALA4033760 | single protein format | Scientific Literature | |
| 19. | ALA4036829 | B | Binding affinity to SK2 (unknown origin) | Homo sapiens | 3 | ALA4033760 | single protein format | Scientific Literature | |
| 20. | ALA4036830 | B | Selectivity ratio of IC50 for human TRPA1 to IC50 for opossum TRPA1 | 1 | ALA4033760 | assay format | Scientific Literature |
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