| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3996975 | F | Agonist activity at human FFA4 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLIPR assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 2. | ALA3996976 | F | Agonist activity at human FFA1 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLIPR assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 3. | ALA3996977 | F | Agonist activity at human FFA4 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLIPR assay relative to GSK137647A | Homo sapiens | 30 | cell-based format | Scientific Literature | ||
| 4. | ALA3996978 | F | Agonist activity at human FFA1 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLIPR assay relative to GSK137647A | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 5. | ALA3996980 | B | Selectivity ratio of EC50 for human FFA1 receptor expressed in human U2OS cells co-expressing Galpha16 to EC50 for human FFA4 receptor expressed in human U2OS cells co-expressing Galpha16 | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 6. | ALA3996982 | A | Clearance in C57BL/6J mouse at 4.2 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 7. | ALA3996984 | A | AUC in C57BL/6J mouse at 4.2 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 8. | ALA3996985 | A | Cmax in C57BL/6J mouse at 10 mg/kg, po | Mus musculus | 5 | organism-based format | Scientific Literature | ||
| 9. | ALA3996986 | A | AUC in C57BL/6J mouse at 10 mg/kg, po | Mus musculus | 5 | organism-based format | Scientific Literature | ||
| 10. | ALA3996987 | A | Oral bioavailability in C57BL/6J mouse at 10 mg/kg | Mus musculus | 5 | organism-based format | Scientific Literature | ||
| 11. | ALA3996988 | A | Half life in C57BL/6J mouse at 10 mg/kg, po | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 12. | ALA3996991 | A | Protein binding in human plasma | Homo sapiens | 5 | cell-free format | Scientific Literature | ||
| 13. | ALA3996992 | B | Agonist activity at mouse FFA4 receptor relative to control | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 14. | ALA3996993 | B | Agonist activity at mouse FFA4 receptor | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 15. | ALA3996994 | B | Agonist activity at rat FFA4 receptor | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 16. | ALA3996995 | B | Agonist activity at rat FFA4 receptor relative to control | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 17. | ALA3996996 | B | Agonist activity at mouse FFA1 receptor | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 18. | ALA3996997 | B | Agonist activity at mouse FFA1 receptor relative to control | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 19. | ALA3996998 | B | Agonist activity at rat FFA1 receptor | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 20. | ALA3996999 | B | Agonist activity at human FFA2 receptor by FLIPR assay | Homo sapiens | 1 | single protein format | Scientific Literature |
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