# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4033874 | F | Antiproliferative activity against human HL60 cells by tryphan blue assay | Homo sapiens | 24 | ALA4033607 | cell-based format | Scientific Literature | |
2. | ALA4151432 | B | Inhibition of GST-tagged human recombinant DYRK1A at 1000 nM by FRET-based LanthaScreen Eu kinase binding assay | Homo sapiens | 17 | ALA4145671 | single protein format | Scientific Literature | |
3. | ALA4151433 | B | Inhibition of GST-tagged human recombinant DYRK1A at 300 nM by FRET-based LanthaScreen Eu kinase binding assay | Homo sapiens | 17 | ALA4145671 | single protein format | Scientific Literature | |
4. | ALA4151434 | B | Inhibition of GST-tagged human recombinant DYRK1A by FRET-based LanthaScreen Eu kinase binding assay | Homo sapiens | 18 | ALA4145671 | single protein format | Scientific Literature | |
5. | ALA4151435 | B | Inhibition of human DYRK1A | Homo sapiens | 2 | ALA4145671 | single protein format | Scientific Literature | |
6. | ALA4151437 | F | Induction of beta-cell proliferation in human pancreatic islets at 10 uM incubated for 96 hrs by Ki67 and insulin immunolabelling method | Homo sapiens | 8 | ALA4145671 | cell-based format | Scientific Literature | |
7. | ALA4151438 | F | Induction of beta-cell proliferation in human pancreatic islets at 30 uM incubated for 96 hrs by Ki67 and insulin immunolabelling method | Homo sapiens | 4 | ALA4145671 | cell-based format | Scientific Literature | |
8. | ALA4151439 | F | Induction of beta-cell proliferation in human pancreatic islets incubated for 96 hrs by Ki67 and insulin immunolabelling method | Homo sapiens | 2 | ALA4145671 | cell-based format | Scientific Literature | |
9. | ALA4151441 | T | Toxicity in human pancreatic islets at 30 uM | Homo sapiens | 2 | ALA4145671 | cell-based format | Scientific Literature | |
10. | ALA4151442 | B | Inhibition of DYRK1A in rat R7T1 cells expressing expressing NFAT2-GFP assessed as induction of NFAT2-GFP nuclear translocation at 10 uM incubated for 24 hrs by | Rattus norvegicus | 2 | ALA4145671 | cell-based format | Scientific Literature | |
11. | ALA4151443 | B | Inhibition of human CDK11 expressed in bacterial expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
12. | ALA4151444 | B | Inhibition of human CDK7 expressed in mammalian expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
13. | ALA4151445 | B | Inhibition of human CDK8 expressed in bacterial expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
14. | ALA4151446 | B | Inhibition of human CDKL5 expressed in mammalian expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
15. | ALA4151447 | B | Inhibition of human CIT expressed in bacterial expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
16. | ALA4151448 | B | Inhibition of human CLK1 expressed in bacterial expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
17. | ALA4151449 | B | Inhibition of human CLK2 expressed in bacterial expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
18. | ALA4151450 | B | Inhibition of human CLK4 expressed in bacterial expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
19. | ALA4151451 | B | Inhibition of human CSNK1A1 expressed in mammalian expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature | |
20. | ALA4151452 | B | Inhibition of human CSNK1D expressed in bacterial expression system assessed as remaining enzyme activity at 10 uM by kinome scan assay | Homo sapiens | 3 | ALA4145671 | assay format | Scientific Literature |