#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4051531	B	Inhibition of His-tagged BRPF1 (626 to 740 residues) (unknown origin) preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,12 diacetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay	Homo sapiens	27		single protein format	Scientific Literature
2.	ALA4051532	B	Inhibition of human BRPF2 (563 to 688 residues) expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,12 diacetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay	Homo sapiens	27		assay format	Scientific Literature
3.	ALA4051533	B	Inhibition of BRPF3 (592 to 711 residues) (unknown origin) preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,12 diacetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay	Homo sapiens	3		single protein format	Scientific Literature
4.	ALA4051534	B	Inhibition of human GST-tagged TAF1 BD2 (1519 to 1651 residues) expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,8,12,16 tetra-acetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay	Homo sapiens	24		assay format	Scientific Literature
5.	ALA4051535	B	Inhibition of human GST-tagged TAF1L BD2 (1517 to 1649 residues) expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,8,12,16 tetra-acetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay	Homo sapiens	3		assay format	Scientific Literature
6.	ALA4051536	B	Inhibition of human BRD4 BD1 (67 to 152 residues) preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,8,12,16 tetra-acetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay	Homo sapiens	27		single protein format	Scientific Literature
7.	ALA4051537	B	Inhibition of BRD4 BD2 (unknown origin) preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,8,12,16 tetra-acetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay	Homo sapiens	27		single protein format	Scientific Literature
8.	ALA4051538	P	Aqueous solubility of the compound in DMSO at pH 6.5 after 24 hrs by HPLC-MS/MS analysis		14		small-molecule physicochemical format	Scientific Literature
9.	ALA4051539	B	Inhibition of Halo-tagged histone H4 binding to C-terminally NanoLuc luciferase conjugated human BRPF2 BD (560 to 666 residues) expressed in human HCT116 cells after 4 to 24 hrs by BRET assay	Homo sapiens	14		cell-based format	Scientific Literature
10.	ALA4051542	B	Inhibition of Halo-tagged histone H4 binding to C-terminally NanoLuc luciferase conjugated BRPF1 BD (626 to 732 residues) (unknown origin) expressed in human HCT116 cells after 4 to 24 hrs by BRET assay	Homo sapiens	5		cell-based format	Scientific Literature
11.	ALA4051593	P	Lipophilicity, log D of the compound at pH 7.5 by reversed-phase HPLC analysis		2		small-molecule physicochemical format	Scientific Literature
12.	ALA4051598	B	Inhibition of Halo-tagged histone H4 binding to C-terminally NanoLuc luciferase conjugated human TAF1 BD2 (1528 to 1640 residues) expressed in human HCT116 cells after 4 to 24 hrs by BRET assay	Homo sapiens	2		cell-based format	Scientific Literature
13.	ALA4051599	A	Apparent permeability across apical to basolateral side in human Caco2 cells at 2 uM after 2 hrs by LC/MS/MS analysis	Homo sapiens	2		cell-based format	Scientific Literature
14.	ALA4051600	A	Apparent permeability across basolateral to apical side in human Caco2 cells at 2 uM after 2 hrs by LC/MS/MS analysis	Homo sapiens	2		cell-based format	Scientific Literature
15.	ALA4051601	A	Efflux ratio of apparent permeability across basolateral to apical over apical to basolateral side in human Caco2 cells at 2 uM after 2 hrs by LC/MS/MS analysis	Homo sapiens	2		cell-based format	Scientific Literature
16.	ALA4051603	B	Inhibition of human BRPF2 (563 to 688 residues) expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 using biotin-acetylated histone H4 peptide as substrate after 30 mins by AlphaScreen assay	Homo sapiens	2		assay format	Scientific Literature
17.	ALA4051604	B	Inhibition of His-tagged BRPF1 (626 to 740 residues) (unknown origin) using biotin-acetylated histone H4 peptide after 30 mins by AlphaScreen assay	Homo sapiens	2		single protein format	Scientific Literature
18.	ALA4051605	B	Inhibition of BRPF3 (592 to 711 residues) (unknown origin) using biotin-acetylated histone H4 peptide as substrate after 30 mins by AlphaScreen assay	Homo sapiens	2		single protein format	Scientific Literature
19.	ALA4051611	B	Inhibition of Halo-tagged histone H3.3 binding to C-terminally NanoLuc luciferase conjugated human BRPF2 BD (560 to 666 residues) expressed in human HCT116 cells after 4 to 24 hrs by BRET assay	Homo sapiens	2		cell-based format	Scientific Literature
20.	ALA4051612	B	Inhibition of Halo-tagged histone H3.3 binding to C-terminally NanoLuc luciferase conjugated human TAF1 BD2 (1528 to 1640 residues) expressed in human HCT116 cells after 4 to 24 hrs by BRET assay	Homo sapiens	2		cell-based format	Scientific Literature