| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4043421 | Binding | Inhibition of recombinant human N-terminal His6-tagged BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) using biotinylated histone peptide as substrate after 60 mins by TR-FRET assay | Homo sapiens | 3 | ALA4043066 | assay format | Scientific Literature | |
| 2. | ALA4043422 | Functional | Antitumor activity against human NCI-H187 cells xenografted subcutaneously in mouse assessed as tumor growth inhibition at 5 mg/kg, po relative to control | Homo sapiens | 1 | ALA4043066 | organism-based format | Scientific Literature |
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