| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4000924 | B | Inhibition of APMA-activated recombinant human MMP-13 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 30 | single protein format | Scientific Literature | ||
| 2. | ALA4000925 | A | Inhibition of APMA-activated recombinant human MMP-2 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 3. | ALA4000926 | A | Inhibition of APMA-activated recombinant human MMP-8 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 4. | ALA4000927 | A | Inhibition of APMA-activated recombinant human MMP-10 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 5. | ALA4000928 | A | Inhibition of CYP3A4 (unknown origin) at 10 uM relative to control | Homo sapiens | 25 | single protein format | Scientific Literature | ||
| 6. | ALA4000929 | A | AUC in rat at 1 mg/kg administered through oral gavage | Rattus norvegicus | 25 | organism-based format | Scientific Literature | ||
| 7. | ALA4000930 | A | Inhibition of APMA-activated recombinant human MMP-1 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 8. | ALA4000931 | A | Inhibition of APMA-activated recombinant human MMP-3 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 9. | ALA4000932 | A | Inhibition of APMA-activated recombinant human MMP-7 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 10. | ALA4000933 | A | Inhibition of APMA-activated recombinant human MMP-9 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 11. | ALA4000934 | A | Inhibition of APMA-activated recombinant human GST-tagged MMP-14 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 12. | ALA4000935 | B | Inhibition of TACE (unknown origin) using Cy3-PLAQAV(Cy5Q-L-2,3-diaminopropionic acid)-RSSSR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 13. | ALA4000936 | U | Selectivity ratio of IC50 for recombinant human MMP-2 to IC50 for human recombinant MMP-13 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 14. | ALA4000937 | U | Selectivity ratio of IC50 for recombinant human MMP-10 to IC50 for human recombinant MMP-13 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 15. | ALA4000938 | U | Selectivity ratio of IC50 for recombinant human MMP-1 to IC50 for human recombinant MMP-13 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 16. | ALA4000939 | U | Selectivity ratio of IC50 for recombinant human MMP-3 to IC50 for human recombinant MMP-13 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 17. | ALA4000940 | U | Selectivity ratio of IC50 for recombinant human MMP-7 to IC50 for human recombinant MMP-13 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 18. | ALA4000941 | U | Selectivity ratio of IC50 for recombinant human MMP-8 to IC50 for human recombinant MMP-13 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 19. | ALA4000942 | U | Selectivity ratio of IC50 for recombinant human MMP-9 to IC50 for human recombinant MMP-13 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 20. | ALA4000943 | U | Selectivity ratio of IC50 for recombinant human GST-tagged MMP-14 to IC50 for human recombinant MMP-13 | Homo sapiens | 2 | assay format | Scientific Literature |
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