| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4009141 | Binding | Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation counting | Cavia porcellus | 26 | ALA4007424 | cell membrane format | Scientific Literature | |
| 2. | ALA4009142 | Binding | Displacement of [3H]DAMGO from mu-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation counting | Cavia porcellus | 16 | ALA4007424 | cell membrane format | Scientific Literature | |
| 3. | ALA4009144 | Binding | Displacement of [3H]DPDPE from delta-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation counting | Cavia porcellus | 25 | ALA4007424 | cell membrane format | Scientific Literature | |
| 4. | ALA4009146 | Binding | Displacement of [3H]-(+)-pentazocine from sigma1-type opioid receptor in guinea pig cortex membranes at 1 uM after 120 mins by solid scintillation counting | Cavia porcellus | 24 | ALA4007424 | cell membrane format | Scientific Literature | |
| 5. | ALA4009148 | Binding | Displacement of [3H]-DTG from sigma 2 receptor in rat liver membranes at 1 uM after 120 mins by scintillation counting | Rattus norvegicus | 23 | ALA4007424 | cell membrane format | Scientific Literature | |
| 6. | ALA4009150 | Binding | Displacement of [3H]-(+)-MK 801 from PCP binding site of NMDA receptor in pig brain cortex membranes at 10 uM after 120 mins by solid scintillation counting | Sus scrofa | 23 | ALA4007424 | cell membrane format | Scientific Literature | |
| 7. | ALA4009152 | Functional | Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assay | Homo sapiens | 25 | ALA4007424 | cell-based format | Scientific Literature | |
| 8. | ALA4009153 | Functional | Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells at 1 uM after 30 mins by [35S]GTPgammaS binding assay | Homo sapiens | 25 | ALA4007424 | cell-based format | Scientific Literature | |
| 9. | ALA4372793 | Binding | Displacement of [3H]U-69,593 from KOR in guinea pig brain membranes after 120 mins by scintillation counting method | Cavia porcellus | 15 | ALA4371059 | cell membrane format | Scientific Literature | |
| 10. | ALA4372795 | Binding | Displacement of [3H]DPDPE from DOR in Sprague-Dawley rat brain membranes after 120 mins by scintillation counting method | Rattus norvegicus | 13 | ALA4371059 | cell membrane format | Scientific Literature | |
| 11. | ALA4372798 | ADME | Displacement of [3H]DAMGO from MOR in guinea pig brain membranes at 1 uM after 120 mins by scintillation counting method relative to control | Cavia porcellus | 13 | ALA4371059 | cell membrane format | Scientific Literature | |
| 12. | ALA4372799 | Binding | Displacement of [3H]DPDPE from DOR in Sprague-Dawley rat brain membranes at 1 uM after 120 mins by scintillation counting method relative to control | Rattus norvegicus | 13 | ALA4371059 | cell membrane format | Scientific Literature | |
| 13. | ALA4372800 | Binding | Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes at 1 uM after 120 mins by scintillation counting method relative to control | Cavia porcellus | 13 | ALA4371059 | cell membrane format | Scientific Literature | |
| 14. | ALA4372801 | Binding | Displacement of [3H]DTG from sigma2 receptor in rat liver membranes at 1 uM after 120 mins by scintillation counting method relative to control | Rattus norvegicus | 13 | ALA4371059 | cell membrane format | Scientific Literature | |
| 15. | ALA4372802 | Binding | Displacement of [3H]diprenorphine from human KOR expressed in HEK293T cell membranes after 120 mins by scintillation counting method | Homo sapiens | 10 | ALA4371059 | cell-based format | Scientific Literature | |
| 16. | ALA4372803 | Functional | Agonist activity at human KOR expressed in HEK293T cells assessed as inhibition of Galphai-mediated cAMP accumulation after 15 mins by microbeta counting assay relative to salvinorin A | Homo sapiens | 9 | ALA4371059 | cell-based format | Scientific Literature | |
| 17. | ALA4372804 | Functional | Agonist activity at human KOR expressed in HEK293T cells assessed as inhibition of Galphai-mediated cAMP accumulation after 15 mins by microbeta counting assay | Homo sapiens | 10 | ALA4371059 | cell-based format | Scientific Literature | |
| 18. | ALA4372805 | Binding | Selectivity ratio of Ki for MOR in guinea pig brain membranes to Ki for KOR in guinea pig brain membranes | Cavia porcellus | 4 | ALA4371059 | cell membrane format | Scientific Literature | |
| 19. | ALA4372806 | Binding | Selectivity ratio of Ki for DOR in Sprague-Dawley rat brain membranes to Ki for KOR in guinea pig brain membranes | 4 | ALA4371059 | cell membrane format | Scientific Literature | ||
| 20. | ALA4372807 | Binding | Selectivity ratio of Ki for sigma1 receptor in guinea pig brain membranes to Ki for KOR in guinea pig brain membranes | Cavia porcellus | 5 | ALA4371059 | cell membrane format | Scientific Literature |
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