| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4029489 | Binding | Inhibition of CDK8 in human SW620 cells assessed as decrease in STAT1 phosphorylation at Ser727 after 2 hrs by Western blot method | Homo sapiens | 36 | ALA4028808 | cell-based format | Scientific Literature | |
| 2. | ALA4029494 | ADME | Intrinsic clearance in human liver microsomes at 1 umol/l after 15 to 30 mins in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 22 | ALA4028808 | assay format | Scientific Literature | |
| 3. | ALA4029551 | Binding | Inhibition of kinase tracer-236 binding to GST-tagged CDK8/CyclinC (unknown origin) after 60 mins by TR-FRET assay | Homo sapiens | 36 | ALA4028808 | protein complex format | Scientific Literature | |
| 4. | ALA4029552 | Binding | Inhibition of kinase tracer-236 binding to GST-tagged CDK19/CyclinC (unknown origin) after 60 mins by TR-FRET assay | Homo sapiens | 36 | ALA4028808 | protein complex format | Scientific Literature |
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