| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4004539 | B | Inhibition of PKCeta (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 2. | ALA4004540 | B | Inhibition of PKCalpha (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 3. | ALA4004541 | B | Inhibition of PKCbeta1 (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 4. | ALA4004542 | B | Inhibition of PKCdelta (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 5. | ALA4004543 | B | Inhibition of PKCepsilon (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 6. | ALA4004544 | B | Inhibition of PKCtheta (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 7. | ALA4004553 | B | Reversible competitive inhibition of PKCalpha (unknown origin) | Homo sapiens | 1 | ALA4002641 | single protein format | Scientific Literature | |
| 8. | ALA4004554 | B | Reversible competitive inhibition of PKCbeta1 (unknown origin) | Homo sapiens | 1 | ALA4002641 | single protein format | Scientific Literature | |
| 9. | ALA4004555 | B | Inhibition of CDK2 (unknown origin) at 1 uM | Homo sapiens | 1 | ALA4002641 | single protein format | Scientific Literature | |
| 10. | ALA4004556 | B | Inhibition of CDK2 (unknown origin) | Homo sapiens | 1 | ALA4002641 | single protein format | Scientific Literature | |
| 11. | ALA4004557 | B | Inhibition of PKCtheta in human Jurkat T cells assessed as reduction in anti-CD3/CD28 antibody-induced T-cell activation by measuring decrease in IL-2 secretion after 5 hrs by luciferase reporter gene assay | Homo sapiens | 6 | ALA4002641 | cell-based format | Scientific Literature | |
| 12. | ALA4004558 | P | Permeability of the compound at pH 6.8 by high-throughput assay | 6 | ALA4002641 | small-molecule physicochemical format | Scientific Literature | ||
| 13. | ALA4004559 | F | Inhibition of human PBMC proliferation assessed as decrease in [3H]-TdR uptake after 6 days by mixed lymphocyte reaction assay | Homo sapiens | 5 | ALA4002641 | cell-based format | Scientific Literature | |
| 14. | ALA4004560 | B | Inhibition of PKCbeta in mouse B cells assessed as reduction in IgM-stimulated cell proliferation | Mus musculus | 2 | ALA4002641 | cell-based format | Scientific Literature | |
| 15. | ALA4004561 | P | Aqueous solubility of the compound | 5 | ALA4002641 | small-molecule physicochemical format | Scientific Literature |
The page will load shortly, Thanks for your patience!