# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4011333 | B | Enhancing of [3H]WIN35,428 binding to recombinant human DAT expressed in HEK293 cell membranes at 10 uM pre-incubated for 10 mins before radioligand addition and measured 90 mins after radioligand addition by micro beta scintillation counting analysis relative to control | Homo sapiens | 20 | ALA4007505 | cell-based format | Scientific Literature | |
2. | ALA4011334 | B | Inhibition of [3H]WIN35,428 binding to recombinant human DAT expressed in HEK293 cell membranes at 10 uM pre-incubated for 10 mins before radioligand addition and measured 90 mins after radioligand addition by micro beta scintillation counting analysis relative to control | Homo sapiens | 20 | ALA4007505 | cell-based format | Scientific Literature | |
3. | ALA4011335 | B | Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from human A3AR expressed in HEK293T cells pre-incubated for 10 mins before radioligand addition and measured 90 mins after radioligand addition by micro beta scintillation counting analysis relative to control | Homo sapiens | 19 | ALA4007505 | cell-based format | Scientific Literature | |
4. | ALA4011337 | B | Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from mouse A3AR expressed in HEK293T cells at 10 uM pre-incubated for 10 mins before radioligand addition and measured 90 mins after radioligand addition by micro beta scintillation counting analysis relative to control | Mus musculus | 14 | ALA4007505 | cell-based format | Scientific Literature | |
5. | ALA4011352 | B | Agonist activity at human A3AR assessed as inhibition of cAMP formation at 10 uM relative to adenosine-5'-Nethyluronamide | Homo sapiens | 3 | ALA4007505 | single protein format | Scientific Literature | |
6. | ALA4011358 | B | Inhibition of [125I]RTI-55 binding to recombinant human SERT expressed in HEK293 cell membranes preincubated for 10 mins followed by radioligand addition measured after 90 mins by micro beta scintillation counting analysis | Homo sapiens | 21 | ALA4007505 | cell-based format | Scientific Literature | |
7. | ALA4011359 | B | Inhibition of [3H]mazindol binding to recombinant human SERT expressed in HEK293 cell membranes preincubated for 10 mins followed by radioligand addition measured after 90 mins by micro beta scintillation counting analysis | Homo sapiens | 22 | ALA4007505 | cell-based format | Scientific Literature | |
8. | ALA4011362 | B | Displacement of [3H]Mesulergine from human 5-HT2C receptor | Homo sapiens | 4 | ALA4007505 | single protein format | Scientific Literature | |
9. | ALA4011366 | B | Displacement of [3H]QNB from human muscarinic M5 receptor | Homo sapiens | 1 | ALA4007505 | single protein format | Scientific Literature | |
10. | ALA4011367 | B | Displacement of [3H]Pentazocine from rat sigma 1 receptor | Rattus norvegicus | 1 | ALA4007505 | single protein format | Scientific Literature | |
11. | ALA4011368 | B | Displacement of [3H]DTG from rat sigma 2 receptor | Rattus norvegicus | 2 | ALA4007505 | single protein format | Scientific Literature |