# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4032440 | B | Displacement of [125I]ABN from human dopamine D3 receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting method | Homo sapiens | 16 | ALA4028897 | cell-based format | Scientific Literature | |
2. | ALA4032441 | B | Displacement of [125I]ABN from human dopamine D2 long receptor expressed in HEK293 cell membranes after 60 mins by scintillation counting method | Homo sapiens | 16 | ALA4028897 | cell-based format | Scientific Literature | |
3. | ALA4032442 | B | Selectivity ratio of Ki for human dopamine D2 long receptor to Ki for human dopamine D3 receptor | Homo sapiens | 15 | ALA4028897 | assay format | Scientific Literature | |
4. | ALA4032443 | B | Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation counting method | Homo sapiens | 4 | ALA4028897 | cell-based format | Scientific Literature | |
5. | ALA4397354 | B | Displacement of [3H]-DAMGO from human MOR stably expressed in HEK cell membranes at 10 uM after 90 mins by microbeta scintillation counting method relative to control | Homo sapiens | 2 | ALA4396871 | cell-based format | Scientific Literature | |
6. | ALA4397355 | B | Displacement of [3H]-DADLE from human DOR stably expressed in HEK cell membranes at 10 uM after 90 mins by microbeta scintillation counting method relative to control | Homo sapiens | 2 | ALA4396871 | cell-based format | Scientific Literature | |
7. | ALA4397356 | B | Displacement of [125I]IABN from recombinant human D3 receptor stably expressed in HEK293 cell membranes measured after 60 mins by scintillation counting analysis | Homo sapiens | 44 | ALA4396871 | cell-based format | Scientific Literature | |
8. | ALA4397357 | A | Displacement of [125I]IABN from recombinant human D2 long receptor stably expressed in HEK293 cell membranes measured after 60 mins by scintillation counting analysis | Homo sapiens | 44 | ALA4396871 | cell-based format | Scientific Literature | |
9. | ALA4397358 | B | Selectivity ratio of Ki for displacement of [125I]IABN from recombinant human D2 long receptor stably expressed in HEK293 cell membranes to Ki for displacement of [125I]IABN from recombinant human D3 receptor stably expressed in HEK293 cell membranes | Homo sapiens | 43 | ALA4396871 | cell-based format | Scientific Literature | |
10. | ALA4397359 | B | Agonist activity at recombinant human D3 receptor expressed in CHOK1 cells assessed as induction of beta arrestin2 recruitment measured after 30 mins by coelenterazine-based beta-galactosidase reporter gene assay | Homo sapiens | 3 | ALA4396871 | cell-based format | Scientific Literature | |
11. | ALA4397360 | A | Antagonist activity at recombinant human D3 receptor expressed in CHOK1 cells assessed as inhibition of dopamine-induced beta arrestin2 recruitment preincubated for 30 mins followed by dopamine addition and measured after 90 mins by coelenterazine-based beta-galactosidase reporter gene assay | Homo sapiens | 3 | ALA4396871 | cell-based format | Scientific Literature | |
12. | ALA4397361 | A | Agonist activity at recombinant human D2 receptor expressed in CHOK1 cells assessed as induction of beta arrestin2 recruitment measured after 30 mins by coelenterazine-based beta-galactosidase reporter gene assay | Homo sapiens | 3 | ALA4396871 | cell-based format | Scientific Literature | |
13. | ALA4397362 | A | Antagonist activity at recombinant human D2 receptor expressed in CHOK1 cells assessed as inhibition of quinpirole-induced beta arrestin2 recruitment preincubated for 30 mins followed by quinpirole addition and measured after 90 mins by coelenterazine-based beta-galactosidase reporter gene assay | Homo sapiens | 3 | ALA4396871 | cell-based format | Scientific Literature | |
14. | ALA4397363 | B | Agonist activity at recombinant human D1 receptor expressed in CHOK1 cells assessed as induction of beta arrestin2 recruitment measured after 30 mins by coelenterazine-based beta-galactosidase reporter gene assay | Homo sapiens | 3 | ALA4396871 | cell-based format | Scientific Literature | |
15. | ALA4397365 | B | Agonist activity at recombinant human D4 receptor expressed in CHOK1 cells assessed as induction of beta arrestin2 recruitment measured after 30 mins by coelenterazine-based beta-galactosidase reporter gene assay | Homo sapiens | 2 | ALA4396871 | cell-based format | Scientific Literature | |
16. | ALA4397368 | B | Displacement of [3H]SCH23390 from recombinant human D1 receptor transiently expressed in HEKT cells at 10 uM measured after 90 mins by microbeta scintillation counting method relative to control | Homo sapiens | 2 | ALA4396871 | cell-based format | Scientific Literature | |
17. | ALA4397370 | B | Displacement of [3H]N-methylspiperone from D3 receptor (unknown origin) measured after 90 mins by microbeta scintillation counting method relative to control | Homo sapiens | 2 | ALA4396871 | single protein format | Scientific Literature | |
18. | ALA4397373 | B | Displacement of [3H]-Way100635 from recombinant human 5HT1A receptor transiently expressed in CHO cell membranes measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 2 | ALA4396871 | cell-based format | Scientific Literature | |
19. | ALA4397375 | B | Displacement of [3H]-5-CT from recombinant human 5HT1B receptor stably expressed in HEK cell membranes measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 1 | ALA4396871 | cell-based format | Scientific Literature | |
20. | ALA4397376 | B | Displacement of [3H]-5-CT from recombinant human 5HT1D receptor transiently expressed in HEKT cell membranes at 10 uM measured after 90 mins by microbeta scintillation counting method relative to control | Homo sapiens | 2 | ALA4396871 | cell-based format | Scientific Literature |