| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4027349 | B | Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation counting method | Rattus norvegicus | 9 | ALA4024770 | assay format | Scientific Literature | |
| 2. | ALA4027350 | B | Displacement of [3H]-AMPA from AMPA receptor in Sprague-Dawley rat brain synaptosomes after 30 mins by scintillation counting method | Rattus norvegicus | 11 | ALA4024770 | subcellular format | Scientific Literature | |
| 3. | ALA4027351 | B | Displacement of [3H]-KA from KA receptor in Sprague-Dawley rat brain synaptosomes after 60 mins by scintillation counting method | Rattus norvegicus | 11 | ALA4024770 | subcellular format | Scientific Literature | |
| 4. | ALA4027352 | B | Displacement of [3H]-CGP-39653 from NMDA receptor in Sprague-Dawley rat brain synaptosomes after 60 mins by scintillation counting method | Rattus norvegicus | 11 | ALA4024770 | subcellular format | Scientific Literature | |
| 5. | ALA4027353 | B | Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation counting method | Rattus norvegicus | 9 | ALA4024770 | assay format | Scientific Literature | |
| 6. | ALA4027354 | B | Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation counting method | Rattus norvegicus | 9 | ALA4024770 | assay format | Scientific Literature | |
| 7. | ALA4027355 | B | Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current responses by two-electrode voltage clamp method | Rattus norvegicus | 2 | ALA4024770 | cell-based format | Scientific Literature | |
| 8. | ALA4027356 | B | Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current responses by two-electrode voltage clamp method | Rattus norvegicus | 2 | ALA4024770 | cell-based format | Scientific Literature | |
| 9. | ALA4027357 | B | Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current responses by two-electrode voltage clamp method | Rattus norvegicus | 2 | ALA4024770 | cell-based format | Scientific Literature | |
| 10. | ALA4027358 | B | Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current responses by two-electrode voltage clamp method | Rattus norvegicus | 2 | ALA4024770 | cell-based format | Scientific Literature | |
| 11. | ALA4027359 | A | AUC (0 to 240 mins) in mouse plasma at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature | |
| 12. | ALA4027360 | A | Cmax in mouse plasma at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature | |
| 13. | ALA4027361 | A | Tmax in mouse plasma at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature | |
| 14. | ALA4027362 | A | Elimination half life in mouse plasma at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature | |
| 15. | ALA4027363 | A | AUC (0 to 240 mins) in mouse liver at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature | |
| 16. | ALA4027364 | A | Cmax in mouse liver at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature | |
| 17. | ALA4027365 | A | Tmax in mouse liver at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature | |
| 18. | ALA4027366 | A | Elimination half life in mouse liver at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature | |
| 19. | ALA4027367 | B | Antagonist activity at NMDA receptor in Nras driven p53 deficient mouse HCC cell membranes assessed as LPS-stimulated PGE2 levels at 10 uM after 24 hrs by LC-MS/MS method (Rvb = 162 +/- 7%) | Mus musculus | 2 | ALA4024770 | assay format | Scientific Literature | |
| 20. | ALA4027368 | A | AUC (0 to 240 mins) in mouse brain at 10 mg/kg, ip administered as bolus dose by LC-MS/MS analysis | Mus musculus | 1 | ALA4024770 | organism-based format | Scientific Literature |
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