| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4005606 | B | Selectivity ratio of IC50 for recombinant G9a catalytic SET domain (913 to 1193 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) codon plus RIL to IC50 for recombinant GLP catalytic SET domain (982 to 1266 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) codon plus RIL | Homo sapiens | 2 | ALA4004823 | assay format | Scientific Literature | |
| 2. | ALA4005607 | B | Inhibition of recombinant GLP catalytic SET domain (982 to 1266 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) codon plus RIL assessed as inhibition of methylation activity using biotin-labeled H3 (1 to 25 residues) as substrate and [3H]-SAM after 2 hrs by scintillation proximity assay | Homo sapiens | 27 | ALA4004823 | assay format | Scientific Literature | |
| 3. | ALA4005608 | B | Inhibition of recombinant G9a catalytic SET domain (913 to 1193 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) codon plus RIL assessed as inhibition of methylation activity using biotin-labeled H3 (1 to 25 residues) as substrate and [3H]-SAM after 2 hrs by scintillation proximity assay | Homo sapiens | 27 | ALA4004823 | assay format | Scientific Literature | |
| 4. | ALA4005637 | B | Inhibition of METTL3-14 (unknown origin) at 10 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 2 | ALA4004823 | protein complex format | Scientific Literature | |
| 5. | ALA4005638 | B | Inhibition of SUV39H1 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 6. | ALA4005639 | B | Inhibition of SUV39H2 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 7. | ALA4005640 | B | Inhibition of SETDB1 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 8. | ALA4005641 | B | Inhibition of SETD7 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 9. | ALA4005642 | B | Inhibition of SETD8 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 10. | ALA4005643 | B | Inhibition of SUV420H1 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 11. | ALA4005644 | B | Inhibition of SUV420H2 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 12. | ALA4005645 | B | Inhibition of MLL1 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 13. | ALA4005646 | B | Inhibition of MLL3 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 14. | ALA4005647 | B | Inhibition of PRDM9 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 15. | ALA4005648 | B | Inhibition of SMYD2 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 16. | ALA4005649 | B | Inhibition of SMYD3 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 17. | ALA4005650 | B | Inhibition of PRC2 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | assay format | Scientific Literature | |
| 18. | ALA4005651 | B | Inhibition of SETD2 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 19. | ALA4005652 | B | Inhibition of PRMT1 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature | |
| 20. | ALA4005653 | B | Inhibition of PRMT3 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | ALA4004823 | single protein format | Scientific Literature |
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