| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4044917 | B | Displacement of [3H]-CGP-12177 from adrenergic beta2 receptor (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA4044918 | B | Displacement of [125I]-(Tyr4)-bombesin from bombesin BB1 receptor (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA4044919 | B | Displacement of [125I]-(Tyr4)-bombesin from bombesin BB2 receptor (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA4044920 | B | Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membranes after 120 mins by liquid scintillation counting | Cavia porcellus | 44 | cell membrane format | Scientific Literature | ||
| 5. | ALA4044923 | B | Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation counting | Rattus norvegicus | 42 | cell membrane format | Scientific Literature | ||
| 6. | ALA4044924 | B | Selectivity index, ratio of Ki for sigma1 receptor in guinea pig brain membranes to Ki for sigma2 receptor in rat liver membranes | 39 | cell membrane format | Scientific Literature | |||
| 7. | ALA4044925 | B | Displacement of [3H]-(+)-MK 801 from PCP binding site of NMDA receptor in pig brain cortex membranes after 120 mins by liquid scintillation spectrometry | Sus scrofa | 39 | cell membrane format | Scientific Literature | ||
| 8. | ALA4044927 | A | Metabolic stability in mouse microsomes assessed as amount of parent compound remaining after 5 mins | Mus musculus | 1 | assay format | Scientific Literature | ||
| 9. | ALA4044928 | A | Metabolic stability in rat microsomes assessed as amount of parent compound remaining after 5 mins | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 10. | ALA4044929 | A | Metabolic stability in human microsomes assessed as amount of parent compound remaining after 5 mins | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA4044930 | A | Inhibition on CYP2C9 (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4044931 | A | Inhibition on CYP2C19 (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4044932 | A | Inhibition on CYP2D6 (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA4044933 | A | Inhibition on CYP3A4 (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA4044934 | A | Binding affinity to human serum albumin at 60 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA4044935 | B | Displacement of [3H]-DPCPX from adenosine A1 receptor (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA4044936 | B | Displacement of [3H]-CGS21680 from adenosine A2A receptor (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA4044937 | B | Displacement of [125I]-AB-MECA from adenosine A3 receptor (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA4044938 | B | Displacement of [3H]-prazosin from adrenergic alpha1A receptor (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4044939 | B | Displacement of [3H]-prazosin from adrenergic alpha1B receptor (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!