| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4011275 | ADME | Stability of compound in Wistar rat brain homogenate assessed as compound remaining at 0.5 mM after 90 mins by RP-HPLC analysis | Rattus norvegicus | 4 | ALA4007500 | tissue-based format | Scientific Literature | |
| 2. | ALA4011276 | Binding | Displacement of [3H]DAMGO from MOR in Wistar rat brain homogenates after 180 mins by liquid scintillation counting analysis | Rattus norvegicus | 4 | ALA4007500 | assay format | Scientific Literature | |
| 3. | ALA4011277 | Binding | Displacement of [3H][Ile5,6]deltorphin-2 from DOR in Wistar rat brain homogenates after 180 mins by liquid scintillation counting analysis | Rattus norvegicus | 4 | ALA4007500 | assay format | Scientific Literature | |
| 4. | ALA4011278 | Binding | Displacement of [3H]nor-BNI from KOR in Dunkin Hartley guinea pig brain homogenates after 180 mins by liquid scintillation counting analysis | Cavia porcellus | 4 | ALA4007500 | assay format | Scientific Literature | |
| 5. | ALA4011280 | Functional | Agonist activity at human recombinant MOR expressed in CHO cells assessed as calcium mobilization by Fluo-4 AM based fluorescence analysis | Homo sapiens | 4 | ALA4007500 | cell-based format | Scientific Literature | |
| 6. | ALA4011281 | Functional | Agonist activity at human recombinant KOR expressed in CHO cells assessed as calcium mobilization up to 1 uM by Fluo-4 AM based fluorescence analysis | Homo sapiens | 3 | ALA4007500 | cell-based format | Scientific Literature | |
| 7. | ALA4011282 | Functional | Agonist activity at human recombinant DOR expressed in CHO cells assessed as calcium mobilization up to 1 uM by Fluo-4 AM based fluorescence analysis | Homo sapiens | 3 | ALA4007500 | cell-based format | Scientific Literature |
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