# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4056671 | B | Inhibition of human GLP catalytic domain (951 to 1235 residues) expressed in Escherichia coli BL21 (DE3) using biotinylated H3 (1 to 25 residues) as substrate preincubated for 20 mins in presence of [3H]SAM measured after 2 hrs by scintillation proximity assay | Homo sapiens | 29 | assay format | Scientific Literature | ||
2. | ALA4056672 | B | Inhibition of human G9a catalytic domain (913 to 1193 residues) expressed in Escherichia coli BL21 (DE3) using biotinylated H3 (1 to 25 residues) as substrate preincubated for 20 mins in presence of [3H]SAM measured after 2 hrs by scintillation proximity assay | Homo sapiens | 29 | assay format | Scientific Literature | ||
3. | ALA4056675 | B | Selectivity ratio of IC50 for human G9a catalytic domain (913 to 1193 residues) to IC50 for human GLP catalytic domain (951 to 1235 residues) | Homo sapiens | 5 | assay format | Scientific Literature |