# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4051803 | Binding | Inhibition of human placental cytosolic 17beta-HSD1 using [3H]-E1/E1 substrate and NADH after 10 mins by HPLC based radio-detection method | Homo sapiens | 13 | ALA4049440 | assay format | Scientific Literature | |
2. | ALA4051804 | ADME | Inhibition of human placental cytosolic 17beta-HSD2 using [3H]-E2/E2 substrate and NAD+ after 20 mins by HPLC based radio-detection method | Homo sapiens | 13 | ALA4049440 | assay format | Scientific Literature | |
3. | ALA4051805 | Unassigned | Selectivity factor, ratio of IC50 for human placental cytosolic 17beta-HSD2 cells to IC50 for human placental cytosolic 17beta-HSD1 | Homo sapiens | 13 | ALA4049440 | assay format | Scientific Literature | |
4. | ALA4051823 | Binding | Inhibition of human placental microsomal STS assessed as formation of E1 at 1 uM preincubated for 30 mins followed by addition of E1S as substrate measured after 20 mins by ELISA | Homo sapiens | 4 | ALA4049440 | assay format | Scientific Literature | |
5. | ALA4051826 | Physicochemical | Stability of the compound in Tris-HCl buffer at pH 7.2 after 30 mins | 10 | ALA4049440 | small-molecule physicochemical format | Scientific Literature |