# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4001326 | B | Inhibition of human EAAT2 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake after 15 mins by TopCount scintillation counting method | Homo sapiens | 4 | ALA4000194 | cell-based format | Scientific Literature | |
2. | ALA4001327 | B | Inhibition of human EAAT3 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake after 15 mins by TopCount scintillation counting method | Homo sapiens | 4 | ALA4000194 | cell-based format | Scientific Literature | |
3. | ALA4001328 | B | Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake after 15 mins by TopCount scintillation counting method | Homo sapiens | 4 | ALA4000194 | cell-based format | Scientific Literature | |
4. | ALA4001329 | B | Displacement of [3H]AMPA from AMPA receptor in rat brain synaptosomal membranes after 30 mins by TopCount microplate scintillation counting method | Rattus norvegicus | 20 | ALA4000194 | cell membrane format | Scientific Literature | |
5. | ALA4001330 | B | Displacement of [3H]kainic acid from kainate receptor in rat brain synaptosomal membranes after 60 mins by TopCount microplate scintillation counting method | Rattus norvegicus | 20 | ALA4000194 | cell membrane format | Scientific Literature | |
6. | ALA4001331 | B | Displacement of [3H]CGP39653 from NMDA receptor in rat brain synaptosomal membranes after 60 mins by TopCount microplate scintillation counting method | Rattus norvegicus | 20 | ALA4000194 | cell membrane format | Scientific Literature | |
7. | ALA4001332 | B | Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting method | Rattus norvegicus | 20 | ALA4000194 | cell-based format | Scientific Literature | |
8. | ALA4001333 | B | Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation counting method | Rattus norvegicus | 20 | ALA4000194 | cell-based format | Scientific Literature | |
9. | ALA4001334 | B | Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation counting method | Rattus norvegicus | 20 | ALA4000194 | cell-based format | Scientific Literature | |
10. | ALA4001335 | B | Antagonist activity at recombinant rat full length GluK1 receptor expressed in HEK293T cells assessed as inhibition of glutamate induced increase in peak current at -100mV holding potential by patch-clamp method | Rattus norvegicus | 1 | ALA4000194 | cell-based format | Scientific Literature | |
11. | ALA4001336 | B | Antagonist activity at recombinant rat full length GluK2 receptor expressed in HEK293T cells assessed as inhibition of glutamate induced increase in peak current at -100mV holding potential by patch-clamp method | Rattus norvegicus | 1 | ALA4000194 | cell-based format | Scientific Literature | |
12. | ALA4001337 | B | Displacement of [3H]-(2S,4R)-4-Methylglutamic acid from rat eGFP-fused GluK1 receptor LBD expressed in HEK293T/17 cells by liquid scintillation counting method | Rattus norvegicus | 1 | ALA4000194 | cell-based format | Scientific Literature |