| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4020427 | B | Inhibition of recombinant human AKR1B10 using pyridine-3-aldehyde as substrate | Homo sapiens | 13 | single protein format | Scientific Literature | ||
| 2. | ALA4020428 | B | Inhibition of recombinant human AKR1B1 using pyridine-3-aldehyde as substrate | Homo sapiens | 13 | single protein format | Scientific Literature | ||
| 3. | ALA4020430 | B | Selectivity ratio of IC50 for recombinant human AKR1B1 to IC50 for recombinant human AKR1B10 | Homo sapiens | 12 | assay format | Scientific Literature | ||
| 4. | ALA4020431 | B | Inhibition of recombinant human AKR1A1 using pyridine-3-aldehyde as substrate | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 5. | ALA4020432 | B | Inhibition of recombinant human AKR1C1 using S-tetralol as substrate | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 6. | ALA4020433 | B | Inhibition of recombinant human AKR1C2 using S-tetralol as substrate | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 7. | ALA4020434 | B | Inhibition of recombinant human AKR1C3 using S-tetralol as substrate | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 8. | ALA4020435 | B | Inhibition of recombinant human AKR1C4 using S-tetralol as substrate | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 9. | ALA4020436 | B | Inhibition of recombinant human CBR1 using isatin as substrate | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 10. | ALA4020437 | B | Selectivity ratio of IC50 for recombinant human AKR1A1 to IC50 for recombinant human AKR1B10 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 11. | ALA4020438 | B | Selectivity ratio of IC50 for recombinant human AKR1C1 to IC50 for recombinant human AKR1B10 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 12. | ALA4020439 | B | Selectivity ratio of IC50 for recombinant human AKR1C2 to IC50 for recombinant human AKR1B10 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 13. | ALA4020440 | B | Selectivity ratio of IC50 for recombinant human AKR1C3 to IC50 for recombinant human AKR1B10 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 14. | ALA4020441 | B | Selectivity ratio of IC50 for recombinant human AKR1C4 to IC50 for recombinant human AKR1B10 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 15. | ALA4020442 | B | Selectivity ratio of IC50 for recombinant human CBR1 to IC50 for recombinant human AKR1B10 | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 16. | ALA4020452 | F | Antimigratory activity in human A549 cells at 20 uM after 24 hrs by wound-healing assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 17. | ALA4020453 | F | Antiproliferative activity against human A549 cells after 96 hrs by tetrazolium-dye based assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 18. | ALA4020454 | F | Antiproliferative activity against human A549/1B10 cells after 96 hrs by tetrazolium-dye based assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 19. | ALA4020455 | F | Antimigratory activity in human A549-Luc2 cells xenografted in C.B-17/IcrHsd-Prkdcscid mouse at 20 uM preincubated for 48 hrs followed by tumor inoculation measured after 4 days by luciferin-based bioluminescence assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 20. | ALA4020456 | F | Antiproliferative activity against human A549/CDDP cells assessed as decrease in cell viability preincubated for 2 hrs followed by addition of 40 uM CDDP addition measured after 24 hrs by tetrazolium-dye based assay | Homo sapiens | 2 | cell-based format | Scientific Literature |
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