| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3995154 | Binding | Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence of NADH by RP-HPLC method | Homo sapiens | 32 | ALA3994586 | assay format | Scientific Literature | |
| 2. | ALA3995155 | Binding | Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method | Homo sapiens | 32 | ALA3994586 | assay format | Scientific Literature | |
| 3. | ALA3995156 | Binding | Selectivity ratio of IC50 for human placental microsomal 17beta-HSD2 to IC50 for human placental cytosolic 17beta-HSD1 | Homo sapiens | 32 | ALA3994586 | assay format | Scientific Literature | |
| 4. | ALA3995157 | ADME | Displacement of [3H]E2 from human recombinant ERalpha assessed as receptor binding at 3 uM after 16 to 20 hrs by liquid scintillation counting method relative to control | Homo sapiens | 8 | ALA3994586 | single protein format | Scientific Literature | |
| 5. | ALA3995158 | ADME | Displacement of [3H]E2 from human recombinant ERbeta assessed as receptor binding at 10 uM after 16 to 20 hrs by liquid scintillation counting method relative to control | Homo sapiens | 8 | ALA3994586 | single protein format | Scientific Literature |
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