| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4015778 | B | Inhibition of SMRT2 H1426W mutant peptide binding to N-terminal His6-tagged human BCL6 BTB domain C8Q/C67R/C84N mutant expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by SMRT2 H1426W mutant peptide addition measured after 60 mins by time-resolved fluorescence resonance energy transfer assay | Homo sapiens | 36 | ALA4014321 | assay format | Scientific Literature | |
| 2. | ALA4015779 | B | Binding affinity to N-terminal His6-tagged human BCL6 BTB domain C8Q/C67R/C84N mutant expressed in Escherichia coli BL21 (DE3) by surface plasmon resonance spectrometry | Homo sapiens | 10 | ALA4014321 | assay format | Scientific Literature | |
| 3. | ALA4015780 | B | Binding affinity to N-terminal His6-tagged human BCL6 BTB domain C8Q/C67R/C84N mutant expressed in Escherichia coli BL21 (DE3) assessed as association rate constant by surface plasmon resonance spectrometry | Homo sapiens | 7 | ALA4014321 | assay format | Scientific Literature | |
| 4. | ALA4015781 | B | Binding affinity to N-terminal His6-tagged human BCL6 BTB domain C8Q/C67R/C84N mutant expressed in Escherichia coli BL21 (DE3) assessed as dissociation rate constant by surface plasmon resonance spectrometry | Homo sapiens | 7 | ALA4014321 | assay format | Scientific Literature | |
| 5. | ALA4015782 | B | Inhibition of human CK2 protein | Homo sapiens | 17 | ALA4014321 | assay format | Scientific Literature | |
| 6. | ALA4015784 | A | Apparent permeability in human Caco2 cells | Homo sapiens | 1 | ALA4014321 | cell-based format | Scientific Literature | |
| 7. | ALA4015786 | P | Aqueous solubility of the compound at pH 7.4 after 24 hrs by LC-UV method | 1 | ALA4014321 | small-molecule physicochemical format | Scientific Literature | ||
| 8. | ALA4015787 | B | Inhibition of GAL4 DNA binding domain fused BCL6 BTB domain (unknown origin) expressed in HEK 293T/17 cells after 24 hrs by Bright-Glo luciferase cell reporter assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 9. | ALA4015788 | B | Inhibition of GAL4 DNA binding domain fused PLZF BTB domain (unknown origin) expressed in HEK 293T/17 cells after 24 hrs by Bright-Glo luciferase cell reporter assay | Homo sapiens | 17 | ALA4014321 | cell-based format | Scientific Literature | |
| 10. | ALA4015789 | F | Antiproliferative activity against BCL6 dependent human OCI-LY1 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 11. | ALA4015790 | F | Antiproliferative activity against BCL6 dependent human TMD8 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 12. | ALA4015791 | F | Antiproliferative activity against BCL6 dependent human OCI-LY3 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 13. | ALA4015792 | F | Antiproliferative activity against BCL6 dependent human OCI-LY10 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 14. | ALA4015793 | F | Antiproliferative activity against BCL6 dependent human SU-DHL-2 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 15. | ALA4015794 | F | Antiproliferative activity against BCL6 dependent human SUDHL4 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 16. | ALA4015795 | F | Antiproliferative activity against BCL6 dependent human U2932 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 17. | ALA4015796 | F | Antiproliferative activity against BCL6 independent human KARPAS422 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 18. | ALA4015797 | F | Antiproliferative activity against BCL6 independent human OCI-LY19 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 19. | ALA4015798 | F | Antiproliferative activity against BCL6 dependent human AMO1 cells after 3 days by CellTiter-Glo assay | Homo sapiens | 18 | ALA4014321 | cell-based format | Scientific Literature | |
| 20. | ALA4015800 | A | Efflux ratio of apparent permeability in human Caco2 cells | Homo sapiens | 1 | ALA4014321 | cell-based format | Scientific Literature |
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