| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4009649 | B | Inhibition of full length His6-tagged PDK1 (unknown origin) expressed in Escherichia coli using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 44 | ALA4007440 | assay format | Scientific Literature | |
| 2. | ALA4009651 | B | Inhibition of PDK2 (unknown origin) using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 4 | ALA4007440 | single protein format | Scientific Literature | |
| 3. | ALA4009652 | B | Inhibition of full length His6-tagged PDK1 (unknown origin) expressed in Escherichia coli assessed as inactivation rate using full length His6-tagged PDHA1 as substrate up to 45 mins by ELISA | Homo sapiens | 10 | ALA4007440 | assay format | Scientific Literature | |
| 4. | ALA4009653 | B | Ratio of Kinact to Ki for full length His6-tagged PDK1 (unknown origin) expressed in Escherichia coli | Homo sapiens | 10 | ALA4007440 | assay format | Scientific Literature | |
| 5. | ALA4009654 | B | Inhibition of PDK1 in human A549 cells assessed as reduction in phosphorylation of PDHE1 at S293 residue at 10 uM after 24 hrs by chemiluminescence/femtochemiluminescence method | Homo sapiens | 11 | ALA4007440 | cell-based format | Scientific Literature | |
| 6. | ALA4009655 | B | Inhibition of PDK1 in human A549 cells assessed as reduction in phosphorylation of PDHE1 at S232 residue at 10 uM after 24 hrs by chemiluminescence/femtochemiluminescence method | Homo sapiens | 9 | ALA4007440 | cell-based format | Scientific Literature | |
| 7. | ALA4009656 | B | Inhibition of PDK1 in human A549 cells assessed as reduction in phosphorylation of PDHE1 at S293 residue at 1 uM after 24 hrs by chemiluminescence/femtochemiluminescence method | Homo sapiens | 9 | ALA4007440 | cell-based format | Scientific Literature | |
| 8. | ALA4009657 | B | Inhibition of PDK1 in human A549 cells assessed as reduction in phosphorylation of PDHE1 at S232 residue at 1 uM after 24 hrs by chemiluminescence/femtochemiluminescence method | Homo sapiens | 9 | ALA4007440 | cell-based format | Scientific Literature | |
| 9. | ALA4009658 | B | Inhibition of PDK1 in human A549 cells assessed as reduction in phosphorylation of PDHE1 at S293 residue after 24 hrs by chemiluminescence/femtochemiluminescence method | Homo sapiens | 3 | ALA4007440 | cell-based format | Scientific Literature | |
| 10. | ALA4009659 | B | Inhibition of PDK1 in human A549 cells assessed as reduction in phosphorylation of PDHE1 at S232 residue after 24 hrs by chemiluminescence/femtochemiluminescence method | Homo sapiens | 3 | ALA4007440 | cell-based format | Scientific Literature | |
| 11. | ALA4009660 | B | Inhibition of PDK2 (unknown origin) assessed as inactivation rate using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 3 | ALA4007440 | single protein format | Scientific Literature | |
| 12. | ALA4009661 | B | Ratio of Kinact to Ki for PDK2 (unknown origin) | Homo sapiens | 3 | ALA4007440 | single protein format | Scientific Literature | |
| 13. | ALA4009662 | B | Inhibition of PDK3 (unknown origin) using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 4 | ALA4007440 | single protein format | Scientific Literature | |
| 14. | ALA4009663 | B | Inhibition of PDK3 (unknown origin) assessed as inactivation rate using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 3 | ALA4007440 | single protein format | Scientific Literature | |
| 15. | ALA4009664 | B | Ratio of Kinact to Ki for PDK3 (unknown origin) | Homo sapiens | 3 | ALA4007440 | single protein format | Scientific Literature | |
| 16. | ALA4009665 | B | Inhibition of full length His6-tagged PDK1 (unknown origin) expressed in Escherichia coli using full length His6-tagged PDHA1 as substrate in presence of GSH after 30 mins by ELISA | Homo sapiens | 4 | ALA4007440 | assay format | Scientific Literature | |
| 17. | ALA4009666 | B | Inhibition of PDK4 (unknown origin) at 10 uM using full length His6-tagged PDHA1 as substrate after 30 mins by ELISA | Homo sapiens | 3 | ALA4007440 | single protein format | Scientific Literature | |
| 18. | ALA4009670 | B | Inhibition of PDK1 in human A549 cells assessed as reduction in extracellular acidification rate after 24 hrs by fluorescent biosensor based assay | Homo sapiens | 3 | ALA4007440 | cell-based format | Scientific Literature | |
| 19. | ALA4009671 | B | Inhibition of PDK1 in human A549 cells assessed as increase in reactive oxygen species after 24 hrs by dihydroethidium staining based FACS analysis | Homo sapiens | 3 | ALA4007440 | cell-based format | Scientific Literature | |
| 20. | ALA4009672 | F | Antiproliferative activity against human A549 cells after 72 hrs by CCK8 assay | Homo sapiens | 4 | ALA4007440 | cell-based format | Scientific Literature |
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