| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4044667 | B | Inhibition of EHMT1 (unknown origin) at 200 uM preincubated for 5 mins followed by SAM and biotinylated H3K9 peptide addition measured after 120 mins by HTRF assay relative to control | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 2. | ALA4044668 | B | Inhibition of EHMT2 (unknown origin) at 400 uM preincubated for 15 mins followed by SAM and biotinylated H3K9 peptide addition measured after 30 mins by TR-FRET assay relative to control | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 3. | ALA4044669 | B | Inhibition of EHMT1 (unknown origin) preincubated for 5 mins followed by SAM and biotinylated H3K9 peptide addition measured after 120 mins by HTRF assay | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 4. | ALA4044670 | B | Inhibition of EHMT2 (unknown origin) preincubated for 15 mins followed by SAM and biotinylated H3K9 peptide addition measured after 30 mins by TR-FRET assay | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 5. | ALA4044671 | B | Inhibition of PRMT1 (unknown origin) at 400 uM preincubated for 5 mins followed by SAM and H4 (1 to 25 residues) peptide addition measured after 1 hr by HTRF assay relative to control | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 6. | ALA4044672 | F | Antiproliferative activity against human HL60 cells at 200 uM after 72 hrs by CCK8 assay relative to control | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 7. | ALA4044673 | F | Antiproliferative activity against human MDA-MB-231 cells at 200 uM after 72 hrs by sulforhodamine B assay relative to control | Homo sapiens | 3 | cell-based format | Scientific Literature |
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