# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4031298 | B | Inhibition of C-terminal His tagged human recombinant HDAC8 (1 to 377 residues) expressed in Baculovirus infected insect cells in presence of ATP | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
2. | ALA4031299 | B | Inhibition of HDAC9 (unknown origin) in presence of ATP | Homo sapiens | 1 | single protein format | Scientific Literature | ||
3. | ALA4031302 | B | Inhibition of C-terminal FLAG His tagged full length human recombinant HDAC1 (1 to 482 residues) expressed in baculovirus infected sf21 cells using RHKKAc as substrate in presence of ATP | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
4. | ALA4031303 | B | Inhibition of C-terminal FLAG His tagged full length human recombinant HDAC1 (1 to 482 residues) expressed in baculovirus infected sf21 cells at 10 uM using RHKKAc as substrate in presence of ATP relative to control | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
5. | ALA4031304 | B | Inhibition of N-terminal GST tagged human HDAC6 (1 to 1215 residues) expressed in baculovirus infected insect cells using RHKKAc as substrate in presence of ATP | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
6. | ALA4031305 | B | Inhibition of human JAK2 using poly[Glu:Tyr] as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 13 | single protein format | Scientific Literature | ||
7. | ALA4031307 | B | Inhibition of human JAK1 using poly[Glu:Tyr] as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 2 | single protein format | Scientific Literature | ||
8. | ALA4031308 | A | Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 2 | single protein format | Scientific Literature | ||
9. | ALA4031309 | B | Inhibition of human TYK2 using KKSRGDYMTMQIG as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 2 | single protein format | Scientific Literature | ||
10. | ALA4031310 | B | Inhibition of human FLT3 using EAIYAAPFAKKK as substrate at 1 uM in presence of [gamma-33P]-ATP relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
11. | ALA4031318 | B | Selectivity ratio of IC50 for human JAK2 to IC50 for human JAK1 | Homo sapiens | 2 | assay format | Scientific Literature | ||
12. | ALA4031319 | U | Selectivity ratio of IC50 for human JAK3 to IC50 for human JAK1 | Homo sapiens | 2 | assay format | Scientific Literature | ||
13. | ALA4031320 | B | Selectivity ratio of IC50 for human TYK2 to IC50 for human JAK1 | Homo sapiens | 2 | assay format | Scientific Literature | ||
14. | ALA4031321 | B | Inhibition of C-terminal GST tagged human recombinant HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells in presence of ATP | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
15. | ALA4031322 | B | Inhibition of human recombinant HDAC3 (1 to 428 residues)/N-terminal GST-tagged NCOR2 (395 to 489 residues) expressed in Baculovirus infected insect cells in presence of ATP | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
16. | ALA4031323 | B | Inhibition of N-terminal GST tagged/C-terminal His tagged human recombinant HDAC4 (627 to 1084 residues) expressed in Baculovirus infected insect cells in presence of ATP | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
17. | ALA4031324 | B | Inhibition of C-terminal His tagged human recombinant HDAC5 (657 to 1123 residues) expressed in Baculovirus infected insect cells in presence of ATP | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
18. | ALA4031326 | B | Inhibition of human HDAC10 using fluorogenic peptide from p53 residues 379 to 382 as substrate in presence of ATP | Homo sapiens | 2 | single protein format | Scientific Literature | ||
19. | ALA4031328 | B | Inhibition of C-terminal His tagged human recombinant HDAC11 (1 to 347 residues) expressed in Baculovirus infected insect cells at 10 uM in presence of ATP relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
20. | ALA4031366 | B | Inhibition of N-terminal GST tagged human HDAC6 (1 to 1215 residues) expressed in baculovirus infected insect cells at 10 uM using RHKKAc as substrate in presence of ATP | Homo sapiens | 13 | cell-based format | Scientific Literature |