| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4018086 | Binding | Inhibition of human coagulation factor 10a | Homo sapiens | 22 | ALA4017471 | single protein format | Scientific Literature | |
| 2. | ALA4018087 | Physicochemical | Apparent permeability of the compound at 5 uM after 5 hrs by PAMPA | 11 | ALA4017471 | small-molecule physicochemical format | Scientific Literature | ||
| 3. | ALA4018088 | Binding | Inhibition of human coagulation factor 9a using SPECTROFLUOR F9a as substrate after 60 mins by fluorescence assay | Homo sapiens | 22 | ALA4017471 | single protein format | Scientific Literature | |
| 4. | ALA4018090 | ADME | Unbound plasma concentration in human at 10 uM measured after 4 hrs by equilibrium dialysis method | Homo sapiens | 11 | ALA4017471 | cell-free format | Scientific Literature | |
| 5. | ALA4018091 | Functional | Anticoagulant activity in human plasma assessed as concentration required to double activated partial thromboplastin time | Homo sapiens | 11 | ALA4017471 | cell-free format | Scientific Literature | |
| 6. | ALA4018094 | Binding | Inhibition of rat coagulation factor 9a | Rattus norvegicus | 1 | ALA4017471 | single protein format | Scientific Literature | |
| 7. | ALA4018095 | Physicochemical | Solubility of the compound in phosphate buffer at pH 7.4 measured after 1.5 hrs by UV absorbance method | 1 | ALA4017471 | small-molecule physicochemical format | Scientific Literature | ||
| 8. | ALA4018096 | ADME | Apparent permeability in MDCK cells at 5 uM after 1 hr by LC-MS/MS method | Canis lupus familiaris | 1 | ALA4017471 | cell-based format | Scientific Literature | |
| 9. | ALA4018097 | ADME | Apparent permeability in MDCK2-MDR1 cells at 5 uM after 1 hr by LC-MS/MS method | Canis lupus familiaris | 1 | ALA4017471 | cell-based format | Scientific Literature | |
| 10. | ALA4018098 | ADME | Metabolic stability in human liver microsomes at 1 uM measured after 20 mins in presence of NADP+ by LC-MS/MS method | Homo sapiens | 1 | ALA4017471 | assay format | Scientific Literature | |
| 11. | ALA4018099 | ADME | Metabolic stability in rat liver microsomes at 1 uM measured after 20 mins in presence of NADP+ by LC-MS/MS method | Rattus norvegicus | 1 | ALA4017471 | assay format | Scientific Literature | |
| 12. | ALA4018100 | ADME | Metabolic stability in dog liver microsomes at 1 uM measured after 20 mins in presence of NADP+ by LC-MS/MS method | Canis lupus familiaris | 1 | ALA4017471 | assay format | Scientific Literature | |
| 13. | ALA4018101 | ADME | Unbound plasma concentration in rat at 10 uM measured after 4 hrs by equilibrium dialysis method | Rattus norvegicus | 1 | ALA4017471 | cell-free format | Scientific Literature | |
| 14. | ALA4018102 | ADME | Unbound plasma concentration in dog at 10 uM measured after 4 hrs by equilibrium dialysis method | Canis lupus familiaris | 1 | ALA4017471 | cell-free format | Scientific Literature | |
| 15. | ALA4018103 | ADME | Volume of distribution at steady state in rat at 1 mg/kg, iv | Rattus norvegicus | 1 | ALA4017471 | organism-based format | Scientific Literature | |
| 16. | ALA4018104 | ADME | Total clearance in rat at 1 mg/kg, iv | Rattus norvegicus | 1 | ALA4017471 | organism-based format | Scientific Literature | |
| 17. | ALA4018105 | ADME | Half life in rat at 1 mg/kg, iv | Rattus norvegicus | 1 | ALA4017471 | organism-based format | Scientific Literature | |
| 18. | ALA4018106 | ADME | AUCt in rat at 1 mg/kg, iv | Rattus norvegicus | 1 | ALA4017471 | organism-based format | Scientific Literature | |
| 19. | ALA4018107 | ADME | Cmax in rat at 10 mg/kg, po | Rattus norvegicus | 1 | ALA4017471 | organism-based format | Scientific Literature | |
| 20. | ALA4018108 | ADME | Tmax in rat at 10 mg/kg, po | Rattus norvegicus | 1 | ALA4017471 | organism-based format | Scientific Literature |
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