| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4023993 | B | Inhibition of fluorescent-labeled 3-(3-((3-(4-amino-5-(4-(3-(2-fluoro-5-(trifluoromethyl)phenyl)ureido)-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)propyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:2',1'-f]-[1,3,2]diazaborinin-4-ium-5-uide binding to human N-terminal GST/His-tagged RIPK1 (1 to 375 residues) expressed in baculovirus expression system by TR-FRET assay | Homo sapiens | 27 | ALA4020836 | assay format | Scientific Literature | |
| 2. | ALA4023995 | B | Inhibition of fluorescent-labeled 3-(3-((3-(4-amino-5-(4-(3-(2-fluoro-5-(trifluoromethyl)phenyl)ureido)-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)propyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:2',1'-f]-[1,3,2]diazaborinin-4-ium-5-uide binding to human N-terminal GST/His-tagged RIPK1 (1 to 375 residues) expressed in baculovirus expression system assessed as association rate constant by TR-FRET assay | Homo sapiens | 26 | ALA4020836 | assay format | Scientific Literature | |
| 3. | ALA4023996 | B | Inhibition of fluorescent-labeled 3-(3-((3-(4-amino-5-(4-(3-(2-fluoro-5-(trifluoromethyl)phenyl)ureido)-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)propyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:2',1'-f]-[1,3,2]diazaborinin-4-ium-5-uide binding to human N-terminal GST/His-tagged RIPK1 (1 to 375 residues) expressed in baculovirus expression system assessed as dissociation rate constant by TR-FRET assay | Homo sapiens | 26 | ALA4020836 | assay format | Scientific Literature | |
| 4. | ALA4023997 | B | Inhibition of fluorescent-labeled 3-(3-((3-(4-amino-5-(4-(3-(2-fluoro-5-(trifluoromethyl)phenyl)ureido)-phenyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)propyl)amino)-3-oxopropyl)-5,5-difluoro-7,9-dimethyl-5H-dipyrrolo[1,2-c:2',1'-f]-[1,3,2]diazaborinin-4-ium-5-uide binding to human N-terminal GST/His-tagged RIPK1 (1 to 375 residues) expressed in baculovirus expression system assessed as dissociation half life by TR-FRET assay | Homo sapiens | 26 | ALA4020836 | assay format | Scientific Literature | |
| 5. | ALA4880779 | B | Adenosine A1 Eurofins-Panlabs radioligand binding assay | Homo sapiens | 20 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 6. | ALA4880780 | B | Adenosine A2A Eurofins-Panlabs radioligand binding assay | Homo sapiens | 20 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 7. | ALA4880781 | B | Adenosine A3 Eurofins-Panlabs radioligand binding assay | Homo sapiens | 16 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 8. | ALA4880784 | B | Adrenergic alpha1D Eurofins-Panlabs radioligand binding assay | Homo sapiens | 13 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 9. | ALA4880785 | B | Adrenergic alpha2A Eurofins-Panlabs radioligand binding assay | Homo sapiens | 12 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 10. | ALA4880786 | B | Adrenergic beta1 Eurofins-Panlabs radioligand binding assay | Homo sapiens | 20 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 11. | ALA4880787 | B | Adrenergic beta2 Eurofins-Panlabs radioligand binding assay | Homo sapiens | 19 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 12. | ALA4880790 | B | Bradykinin B2 Eurofins-Panlabs radioligand binding assay | Homo sapiens | 11 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 13. | ALA4880791 | B | Calcium Channel L-Type, Benzothiazepine Eurofins-Panlabs radioligand binding assay | Rattus sp. | 13 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 14. | ALA4880792 | B | Calcium Channel L-Type, Dihydropyridine Eurofins-Panlabs radioligand binding assay | Rattus sp. | 13 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 15. | ALA4880793 | B | Calcium Channel N-Type Eurofins-Panlabs radioligand binding assay | Rattus sp. | 12 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 16. | ALA4880795 | B | Dopamine D1 Eurofins-Panlabs radioligand binding assay | Homo sapiens | 21 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 17. | ALA4880796 | B | Dopamine D2S Eurofins-Panlabs radioligand binding assay | Homo sapiens | 18 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 18. | ALA4880797 | B | Dopamine D3 Eurofins-Panlabs radioligand binding assay | Homo sapiens | 17 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 19. | ALA4880799 | B | Endothelin ETA Eurofins-Panlabs radioligand binding assay | Homo sapiens | 18 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt | |
| 20. | ALA4880800 | B | Endothelin ETB Eurofins-Panlabs radioligand binding assay | Homo sapiens | 17 | ALA4507332 | single protein format | Donated Chemical Probes - SGC Frankfurt |
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