| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4040374 | Binding | Inhibition of recombinant human N-terminal GST-tagged ROCK2 catalytic domain (1 to 553 residues) expressed in baculovirus expression system using STK 2-biotin as substrate measured after 60 mins by HTRF/TR-FRET assay | Homo sapiens | 92 | ALA4038320 | assay format | Scientific Literature | |
| 2. | ALA4040375 | Binding | Inhibition of recombinant human N-terminal GST-tagged GRK2 expressed in baculovirus expression system using ulight topo2alpha as substrate preincubated for 60 mins followed by substrate addition measured after 10 mins by Lance TR-FRET assay | Homo sapiens | 92 | ALA4038320 | assay format | Scientific Literature | |
| 3. | ALA4040376 | Binding | Inhibition of human PKCalpha active using MBP as substrate after 60 mins in presence of [gamma-32]ATP by scintillation counting | Homo sapiens | 92 | ALA4038320 | single protein format | Scientific Literature | |
| 4. | ALA4040377 | ADME | Inhibition of CYP3A4 (unknown origin) at 10 uM | Homo sapiens | 78 | ALA4038320 | single protein format | Scientific Literature |
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