| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4014035 | B | Inhibition of PDE5A1 catalytic domain (535 to 860 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using [3H]cGMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 22 | ALA4011656 | assay format | Scientific Literature | |
| 2. | ALA4014036 | A | Half life in Sprague-Dawley rat at 5 mg/kg, po by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 3. | ALA4014037 | A | Half life in Sprague-Dawley rat at 2.5 mg/kg, iv by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 4. | ALA4014038 | A | Tmax in Sprague-Dawley rat at 5 mg/kg, po by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 5. | ALA4014039 | A | Cmax in Sprague-Dawley rat at 5 mg/kg, po by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 6. | ALA4014040 | A | Cmax in Sprague-Dawley rat at 2.5 mg/kg, iv by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 7. | ALA4014041 | A | AUC (0 to t) in Sprague-Dawley rat at 5 mg/kg, po by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 8. | ALA4014042 | A | AUC (0 to t) in Sprague-Dawley rat at 2.5 mg/kg, iv by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 9. | ALA4014043 | A | AUC (0 to infinity) in Sprague-Dawley rat at 5 mg/kg, po by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 10. | ALA4014044 | A | AUC (0 to infinity) in Sprague-Dawley rat at 2.5 mg/kg, iv by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 11. | ALA4014045 | A | MRT (0 to t) in Sprague-Dawley rat at 5 mg/kg, po by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 12. | ALA4014046 | A | MRT (0 to t) in Sprague-Dawley rat at 2.5 mg/kg, iv by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 13. | ALA4014047 | A | Oral bioavailability in Sprague-Dawley rat at 5 mg/kg by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA4011656 | organism-based format | Scientific Literature | |
| 14. | ALA4014050 | B | Inhibition of PDE1B (10 to 487 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using [3H]cAMP or [3H]cGMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 1 | ALA4011656 | assay format | Scientific Literature | |
| 15. | ALA4014051 | B | Inhibition of PDE2A (580 to 919 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using [3H]cGMP or [3H]cAMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 1 | ALA4011656 | assay format | Scientific Literature | |
| 16. | ALA4014052 | B | Inhibition of PDE3A (679 to 1087 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using [3H]cAMP or [3H]cGMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 1 | ALA4011656 | assay format | Scientific Literature | |
| 17. | ALA4014053 | B | Inhibition of PDE4D2 (86 to 413 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using [3H]cAMP or [3H]cGMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 1 | ALA4011656 | assay format | Scientific Literature | |
| 18. | ALA4014054 | B | Inhibition of PDE6A (484 to 817 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using [3H]cGMP or [3H]cAMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 1 | ALA4011656 | assay format | Scientific Literature | |
| 19. | ALA4014055 | B | Inhibition of PDE7A1 (130 to 482 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using [3H]cGMP or [3H]cAMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 1 | ALA4011656 | assay format | Scientific Literature | |
| 20. | ALA4014056 | B | Inhibition of PDE8A1 (480 to 820 residues) (unknown origin) using [3H]cGMP or [3H]cAMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 1 | ALA4011656 | single protein format | Scientific Literature |
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