| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4004539 | Binding | Inhibition of PKCeta (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 2. | ALA4004540 | Binding | Inhibition of PKCalpha (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 3. | ALA4004541 | Binding | Inhibition of PKCbeta1 (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 4. | ALA4004542 | Binding | Inhibition of PKCdelta (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 5. | ALA4004543 | Binding | Inhibition of PKCepsilon (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 6. | ALA4004544 | Binding | Inhibition of PKCtheta (unknown origin) after 60 mins in presence of [gamma33P]ATP by scintillation proximity assay | Homo sapiens | 18 | ALA4002641 | single protein format | Scientific Literature | |
| 7. | ALA4004545 | Binding | Ratio of IC50 for PKCdelta (unknown origin) to IC50 for PKCalpha (unknown origin) | Homo sapiens | 1 | ALA4002641 | assay format | Scientific Literature | |
| 8. | ALA4004546 | Binding | Ratio of IC50 for PKCepsilon (unknown origin) to IC50 for PKCalpha (unknown origin) | Homo sapiens | 1 | ALA4002641 | assay format | Scientific Literature | |
| 9. | ALA4004547 | Binding | Ratio of IC50 for PKCeta (unknown origin) to IC50 for PKCalpha (unknown origin) | Homo sapiens | 1 | ALA4002641 | assay format | Scientific Literature | |
| 10. | ALA4004548 | Binding | Ratio of IC50 for PKCtheta (unknown origin) to IC50 for PKCalpha (unknown origin) | Homo sapiens | 1 | ALA4002641 | assay format | Scientific Literature | |
| 11. | ALA4004549 | Binding | Ratio of IC50 for PKCdelta (unknown origin) to IC50 for PKCbeta1 (unknown origin) | Homo sapiens | 1 | ALA4002641 | assay format | Scientific Literature | |
| 12. | ALA4004550 | Binding | Ratio of IC50 for PKCepsilon (unknown origin) to IC50 for PKCbeta1 (unknown origin) | Homo sapiens | 1 | ALA4002641 | assay format | Scientific Literature | |
| 13. | ALA4004551 | Binding | Ratio of IC50 for PKCeta (unknown origin) to IC50 for PKCbeta1 (unknown origin) | Homo sapiens | 1 | ALA4002641 | assay format | Scientific Literature | |
| 14. | ALA4004552 | Binding | Ratio of IC50 for PKCtheta (unknown origin) to IC50 for PKCbeta1 (unknown origin) | Homo sapiens | 1 | ALA4002641 | assay format | Scientific Literature | |
| 15. | ALA4004557 | Binding | Inhibition of PKCtheta in human Jurkat T cells assessed as reduction in anti-CD3/CD28 antibody-induced T-cell activation by measuring decrease in IL-2 secretion after 5 hrs by luciferase reporter gene assay | Homo sapiens | 6 | ALA4002641 | cell-based format | Scientific Literature | |
| 16. | ALA4004558 | Physicochemical | Permeability of the compound at pH 6.8 by high-throughput assay | 6 | ALA4002641 | small-molecule physicochemical format | Scientific Literature | ||
| 17. | ALA4004559 | Functional | Inhibition of human PBMC proliferation assessed as decrease in [3H]-TdR uptake after 6 days by mixed lymphocyte reaction assay | Homo sapiens | 5 | ALA4002641 | cell-based format | Scientific Literature | |
| 18. | ALA4004561 | Physicochemical | Aqueous solubility of the compound | 5 | ALA4002641 | small-molecule physicochemical format | Scientific Literature |
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