# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4019582 | B | Irreversible inhibition of human TG2 using AL5 as substrate by colorimetric assay | Homo sapiens | 27 | ALA4017513 | single protein format | Scientific Literature | |
2. | ALA4019583 | B | Ratio of kinact to Ki for human TG2 by by colorimetric assay | Homo sapiens | 27 | ALA4017513 | single protein format | Scientific Literature | |
3. | ALA4019584 | B | Inhibition of human TG2 binding with BODIPY GTP-gamma-S preincubated for 30 mins followed by BODIPY GTP-gamma-S addition measured after 10 mins | Homo sapiens | 2 | ALA4017513 | single protein format | Scientific Literature | |
4. | ALA4019585 | B | Inactivation of human TG1 using AL5 as substrate by colorimetric assay | Homo sapiens | 2 | ALA4017513 | single protein format | Scientific Literature | |
5. | ALA4019586 | B | Inactivation of human F13a assessed as rate constant of enzyme inhibition using FRET- quenched A101 as substrate by fluorescence assay | Homo sapiens | 2 | ALA4017513 | single protein format | Scientific Literature | |
6. | ALA4019587 | B | Inactivation of activated human TG3 assessed as rate constant of enzyme inactivation using FRET- quenched A101 as substrate by fluorescence assay | Homo sapiens | 2 | ALA4017513 | single protein format | Scientific Literature | |
7. | ALA4019588 | B | Inactivation of human TG6 using AL5 as substrate by colorimetric assay | Homo sapiens | 2 | ALA4017513 | single protein format | Scientific Literature | |
8. | ALA4019589 | F | Inhibition of human ECS cells invasion by using Engelbreth-Holm-Swarm mouse tumor matrigel measured after 18 hrs by DAPI staining-based flourescence microscopy | Homo sapiens | 2 | ALA4017513 | cell-based format | Scientific Literature | |
9. | ALA4019595 | B | Selectivity ratio of Kobs for human TG2 to Kobs for activated human TG3 | Homo sapiens | 2 | ALA4017513 | assay format | Scientific Literature | |
10. | ALA4019596 | B | Selectivity ratio of Kobs for human TG2 to Kobs for human TG1 | Homo sapiens | 1 | ALA4017513 | assay format | Scientific Literature | |
11. | ALA4019597 | B | Selectivity ratio of Kobs for human TG2 to Kobs for human F13a | Homo sapiens | 1 | ALA4017513 | assay format | Scientific Literature | |
12. | ALA5158929 | B | Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate assessed as Kinact/Ki ratio and measured by colorimetric assay | Homo sapiens | 46 | ALA5154739 | single protein format | Scientific Literature | |
13. | ALA5158930 | B | Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assay | Homo sapiens | 47 | ALA5154739 | single protein format | Scientific Literature | |
14. | ALA5158948 | F | Anti-invasion activity against human SCC-13 cells assessed as inhibition of invasion incubated for 18 hrs by matrigel trans well plate assay | Homo sapiens | 6 | ALA5154739 | cell-based format | Scientific Literature |