#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4050596	B	Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mins by spectrofluorometry method	Homo sapiens	75	ALA4049407	cell-based format	Scientific Literature
2.	ALA4050597	B	Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mins by spectrofluorometry method	Homo sapiens	75	ALA4049407	cell-based format	Scientific Literature
3.	ALA4050598	B	Selectivity index, ratio of Ki for recombinant human furin expressed in drosophila S2 cells to Ki for recombinant human PACE4 expressed in drosophila S2 cells	Homo sapiens	75	ALA4049407	cell-based format	Scientific Literature
4.	ALA4050600	F	Antiproliferative activity against human DU145 cells assessed as reduction in metabolic activity after 72 hrs by MTT assay	Homo sapiens	23	ALA4049407	cell-based format	Scientific Literature
5.	ALA4050601	F	Antiproliferative activity against human LNCAP cells assessed as reduction in metabolic activity after 72 hrs by MTT assay	Homo sapiens	23	ALA4049407	cell-based format	Scientific Literature
6.	ALA4236725	F	Antitumor activity against human LNCAP cells xenografted in nu mouse assessed as reduction in tumor volume at 2 mg/kg/day, iv administered at 24 hr intervals	Homo sapiens	1	ALA4229560	organism-based format	Scientific Literature
7.	ALA4236726	F	Antitumor activity against human LNCAP cells xenografted in nu mouse assessed as reduction in serum prostate-specific antigen levels at 2 mg/kg/day, iv administered at 24 hr intervals	Homo sapiens	1	ALA4229560	organism-based format	Scientific Literature
8.	ALA4236727	B	Inhibition of recombinant human PACE4 expressed in S2 insect cells using pyroGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate after 1 hr by spectrofluorometry	Homo sapiens	27	ALA4229560	cell-based format	Scientific Literature
9.	ALA4236728	T	Acute toxicity in iv dosed CD1 mouse measured within 5 mins post dose	Mus musculus	1	ALA4229560	organism-based format	Scientific Literature
10.	ALA4236729	A	Half life in human plasma by ion chromatogram-based analysis	Homo sapiens	3	ALA4229560	cell-free format	Scientific Literature
11.	ALA4236736	F	Antiproliferative activity against human DU145 cells after 72 hrs by MTT assay	Homo sapiens	23	ALA4229560	cell-based format	Scientific Literature
12.	ALA4236737	F	Antiproliferative activity against human LNCAP cells after 72 hrs by MTT assay	Homo sapiens	25	ALA4229560	cell-based format	Scientific Literature
13.	ALA4236738	B	Selectivity ratio of Ki for recombinant human furin to Ki for recombinant human PACE4	Homo sapiens	27	ALA4229560	assay format	Scientific Literature
14.	ALA4236739	B	Inhibition of recombinant human furin expressed in S2 insect cells using pyroGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate after 1 hr by spectrofluorometry	Homo sapiens	27	ALA4229560	cell-based format	Scientific Literature
15.	ALA4261461	B	Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometry	Homo sapiens	12	ALA4257595	single protein format	Scientific Literature
16.	ALA4261462	B	Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometry	Homo sapiens	12	ALA4257595	single protein format	Scientific Literature
17.	ALA4261463	B	Selectivity ratio of Ki for recombinant human furin to Ki for recombinant human PACE4	Homo sapiens	12	ALA4257595	assay format	Scientific Literature
18.	ALA4261464	F	Antiproliferative activity against human DU145 cells after 72 hrs by MTT assay	Homo sapiens	12	ALA4257595	cell-based format	Scientific Literature
19.	ALA4261465	F	Antiproliferative activity against human LNCAP cells after 72 hrs by MTT assay	Homo sapiens	12	ALA4257595	cell-based format	Scientific Literature