# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4043777 | B | Inhibition of human recombinant His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus using Tyr-4 peptide after 1 hr by FRET-based Z'-Lyte assay | Homo sapiens | 23 | ALA4043093 | assay format | Scientific Literature | |
2. | ALA4043778 | B | Inhibition of human recombinant cytoplasmic His-tagged FGFR2 (403 to 822 residues) expressed in baculovirus using Tyr-4 peptide after 1 hr by FRET-based Z'-Lyte assay | Homo sapiens | 14 | ALA4043093 | assay format | Scientific Literature | |
3. | ALA4043779 | B | Inhibition of human recombinant His-tagged FGFR3 cytoplasmic domain (399 to 806 residues) expressed in baculovirus using Tyr-4 peptide after 1 hr by FRET-based Z'-Lyte assay | Homo sapiens | 14 | ALA4043093 | assay format | Scientific Literature | |
4. | ALA4043780 | B | Inhibition of human recombinant His-tagged FGFR4 cytoplasmic domain (781 to 1338 residues) expressed in baculovirus using Tyr-4 peptide after 1 hr by FRET-based Z'-Lyte assay | Homo sapiens | 14 | ALA4043093 | assay format | Scientific Literature | |
5. | ALA4043781 | F | Antiproliferative activity against human FGFR1-amplified NCI-H520 cells after 7 days by SRB assay | Homo sapiens | 15 | ALA4043093 | cell-based format | Scientific Literature | |
6. | ALA4043782 | F | Antiproliferative activity against human FGFR3-amplified SW780 cells after 5 days by SRB assay | Homo sapiens | 15 | ALA4043093 | cell-based format | Scientific Literature | |
7. | ALA4043792 | F | Antiproliferative activity against human FGFR2-amplified SUM52 cells after 5 days by SRB assay | Homo sapiens | 15 | ALA4043093 | cell-based format | Scientific Literature |