| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4122970 | B | Displacement of H3K4me3 binding to Halo-tagged GST-fused KDM5A PHD3 domain (unknown origin) expressed in Escherichia coli by HaloTag-based peptide displacement assay | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 2. | ALA4122971 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from recombinant His6-tagged human KDM5A (PHD3) (1542 to 1660 residues) expressed in Escherichia coli 2(DE3)pLysS Rosetta competent cells preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 18 | cell-based format | Scientific Literature | ||
| 3. | ALA4122975 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 15 | single protein format | Scientific Literature | ||
| 4. | ALA4122976 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7B (PHD) (unknown origin) preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 15 | single protein format | Scientific Literature | ||
| 5. | ALA4122977 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7C (PHD) (unknown origin) preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 15 | single protein format | Scientific Literature | ||
| 6. | ALA4122978 | B | Binding affinity to biotin-His6 peptide (unknown origin) by counterscreen assay | Not specified | 12 | assay format | Scientific Literature | ||
| 7. | ALA4122980 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) at 100 uM preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4122981 | B | Inhibition of KDM7A (PHD-JmjC) (unknown origin) demethylation activity at 100 uM preincubated for 10 mins followed by H3(1-15)K9me2 peptide substrate addition by MALDI-TOF-MS analysis | Homo sapiens | 7 | single protein format | Scientific Literature | ||
| 9. | ALA4122983 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7B (PHD-JmjC) (unknown origin) at 100 uM preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 10. | ALA4122984 | B | Inhibition of KDM7B (PHD-JmjC) (unknown origin) demethylation activity at 100 uM preincubated for 10 mins followed by H3(1-15)K4me3K9me2 peptide substrate addition by MALDI-TOF-MS analysis | Homo sapiens | 7 | single protein format | Scientific Literature | ||
| 11. | ALA4138817 | B | Inhibition of recombinant HQ5-Halo-tagged JARID1A PHD3 finger domain (unknown origin) expressed in BL21(DE3)pLysS cells after 1 hr by chemiluminescent assay | Homo sapiens | 2 | cell-based format | Scientific Literature |
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