| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4124800 | F | Agonist activity at human GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Homo sapiens | 16 | ALA4118251 | cell-based format | Scientific Literature | |
| 2. | ALA4124801 | F | Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Homo sapiens | 16 | ALA4118251 | cell-based format | Scientific Literature | |
| 3. | ALA4124802 | F | Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Homo sapiens | 16 | ALA4118251 | cell-based format | Scientific Literature | |
| 4. | ALA4124810 | B | Agonist activity at monkey GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Macaca mulatta | 4 | ALA4118251 | cell-based format | Scientific Literature | |
| 5. | ALA4124811 | B | Agonist activity at monkey glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Macaca mulatta | 4 | ALA4118251 | cell-based format | Scientific Literature | |
| 6. | ALA4124812 | B | Agonist activity at monkey GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Macaca mulatta | 4 | ALA4118251 | cell-based format | Scientific Literature | |
| 7. | ALA4378455 | A | Half life in human plasma | Homo sapiens | 1 | ALA4376821 | cell-free format | Scientific Literature | |
| 8. | ALA4673578 | A | Half life in iv dosed Wistar rat serum measured after 2 to 20 mins by HPLC analysis | Rattus norvegicus | 1 | ALA4673185 | organism-based format | Scientific Literature | |
| 9. | ALA4704626 | F | Hypoglycemic activity in ICR mouse assessed as decrease in blood glucose concentration at 25 nmol/kg, ip dosed 15 mins before test and measured up to 120 mins by OGTT method | Mus musculus | 10 | ALA4699602 | organism-based format | Scientific Literature | |
| 10. | ALA5245917 | B | Agonist activity at mouse GLP-1R expressed in CHO cells assessed as increase in cAMP accumulation | Mus musculus | 11 | ALA5244248 | cell-based format | Scientific Literature | |
| 11. | ALA5245920 | F | Anti-apoptotic activity in rat INS1 cells assessed as reduction in cytokine-induced cell apoptosis at 100 nM treated for 1 hr prior to TNF-alpha and IL-1beta challenge | Rattus norvegicus | 2 | ALA5244248 | cell-based format | Scientific Literature |
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