#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4121347	B	Binding affinity to recombinant human RORgamma LBD (237 to 497 residues) expressed in Escherichia coli BL21 (DE3) GOLD by 1,8-ANS dye-based thermofluor assay	Homo sapiens	48	ALA4118122	assay format	Scientific Literature
2.	ALA4121348	B	Binding affinity to recombinant human RORbeta LBD (201 to 452 residues) expressed in Escherichia coli BL21 (DE3) GOLD by 1,8-ANS dye-based thermofluor assay	Homo sapiens	47	ALA4118122	assay format	Scientific Literature
3.	ALA4121349	B	Inverse agonist activity at human GAL4 DBD-fused RORgammat LBD (237 to 497 residues) expressed in HEK293T cells assessed as reduction in ROR mediated transcriptional activity after 24 hrs by dual glo luciferase reporter gene assay	Homo sapiens	49	ALA4118122	cell-based format	Scientific Literature
4.	ALA4121350	B	Inverse agonist activity at human GAL4 DBD-fused RORgammat LBD (237 to 497 residues) expressed in HEK293T cells assessed as reduction in ROR mediated transcriptional activity after 24 hrs by dual glo luciferase reporter gene assay relative to T0901317	Homo sapiens	49	ALA4118122	cell-based format	Scientific Literature
5.	ALA4121351	B	Inverse agonist activity at human GAL4 DBD-fused RORbeta LBD (201 to 452 residues) expressed in HEK293T cells assessed as reduction in ROR mediated transcriptional activity after 24 hrs by dual glo luciferase reporter gene assay	Homo sapiens	23	ALA4118122	cell-based format	Scientific Literature
6.	ALA4121352	B	Inverse agonist activity at human GAL4 DBD-fused RORbeta LBD (201 to 452 residues) expressed in HEK293T cells assessed as reduction in ROR mediated transcriptional activity after 24 hrs by dual glo luciferase reporter gene assay relative to N-[5-(2-chloro-benzoyl)-4-(3-chlorophenyl)-thiazol-2-yl]-2-(4-ethanesulfonyl-phenyl)-acetamide	Homo sapiens	17	ALA4118122	cell-based format	Scientific Literature
7.	ALA4121353	B	Inverse agonist activity at RORgammat in human CD4 positive T cells assessed as inhibition of IL17A production in human Th17 cells after 1 hr	Homo sapiens	17	ALA4118122	cell-based format	Scientific Literature
8.	ALA4121356	B	Inverse agonist activity at RORgammat in human CD4 positive T cells assessed as inhibition of IL17A production in human Th17 cells at 0.2 uM after 1 hr relative to JNJ-54271074	Homo sapiens	1	ALA4118122	cell-based format	Scientific Literature
9.	ALA4121357	A	Inverse agonist activity at PXR LBD (unknown origin) expressed in HEK293 cells assessed as decrease in PXR mediated transcriptional activity at 1 uM after 16 hrs by luciferase reporter gene assay relative to rifampicin	Homo sapiens	39	ALA4118122	cell-based format	Scientific Literature
10.	ALA4121359	B	Inverse agonist activity at RORgammat in human whole blood assessed as reduction in IL17A production	Homo sapiens	28	ALA4118122	single protein format	Scientific Literature
11.	ALA4121360	B	Inverse agonist activity at RORgammat in human whole blood assessed as reduction in IL17A production at 1 uM relative to JNJ-54271074	Homo sapiens	25	ALA4118122	single protein format	Scientific Literature
12.	ALA4121361	B	Displacement of [3H]-DPCPX from human recombinant adenosine A1 receptor at 10 uM after 60 mins by scintillation counting analysis relative to control	Homo sapiens	1	ALA4118122	single protein format	Scientific Literature
13.	ALA4121362	B	Displacement of [3H]-CGS 21680 from human recombinant adenosine A2A receptor at 10 uM after 120 mins by scintillation counting analysis relative to control	Homo sapiens	1	ALA4118122	single protein format	Scientific Literature
14.	ALA4121363	B	Displacement of [125I]AB-MECA from human recombinant adenosine A3 receptor at 10 uM after 120 mins by scintillation counting analysis relative to control	Homo sapiens	1	ALA4118122	single protein format	Scientific Literature
15.	ALA4121364	B	Displacement of [3H]-prazosin from rat alpha1 adrenoceptor at 10 uM after 60 mins by scintillation counting analysis relative to control	Rattus norvegicus	1	ALA4118122	protein format	Scientific Literature
16.	ALA4121365	B	Displacement of [3H]-RX 821002 from rat alpha2 adrenoceptor at 10 uM after 60 mins by scintillation counting analysis relative to control	Rattus norvegicus	1	ALA4118122	protein format	Scientific Literature
17.	ALA4121366	B	Displacement of [3H](-)CGP 12177 from human beta1 adrenoceptor at 10 uM after 60 mins by scintillation counting analysis relative to control	Homo sapiens	1	ALA4118122	single protein format	Scientific Literature
18.	ALA4121367	B	Displacement of [125I][Sar1,Ile8]-AT-II from human recombinant AT1 receptor at 10 uM after 120 mins by scintillation counting analysis relative to control	Homo sapiens	1	ALA4118122	single protein format	Scientific Literature
19.	ALA4121368	B	Displacement of [3H]flunitrazepam from rat brain central BZD at 10 uM after 60 mins relative to control	Rattus norvegicus	1	ALA4118122	assay format	Scientific Literature
20.	ALA4121369	B	Displacement of [3H]bradykinin from human recombinant B2 receptor at 10 uM after 60 mins by scintillation counting analysis relative to control	Homo sapiens	1	ALA4118122	single protein format	Scientific Literature