| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4120238 | B | Inhibition of PKC-delta (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 2. | ALA4120241 | F | Antiinflammatory activity in C57BL/6J mouse assessed as reduction in recombinant mouse IL-6 induced serum hepcidin level at 30 mg/kg, po pretreated for 30 mins followed by IL-6 challenge and measured after 4 hrs by LC-MS/MS analysis | Mus musculus | 1 | ALA4118098 | organism-based format | Scientific Literature | |
| 3. | ALA4120242 | F | Inhibition of human recombinant BMP6-stimulated hepcidin mRNA expression in human HepG2 cells after 6 hrs by qRT-PCR analysis | Homo sapiens | 28 | ALA4118098 | cell-based format | Scientific Literature | |
| 4. | ALA4120243 | A | Metabolic stability in pooled CD1 mouse liver microsomes assessed as parent compound remaining at 1 uM after 30 mins by LC-MS/MS analysis | Mus musculus | 1 | ALA4118098 | microsome format | Scientific Literature | |
| 5. | ALA4120244 | A | Fraction unbound in mouse plasma | Mus musculus | 1 | ALA4118098 | cell-free format | Scientific Literature | |
| 6. | ALA4120245 | P | Lipophilicity, log D of the compound | 1 | ALA4118098 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA4120246 | A | Cmax in C57BL/6J mouse at 30 mg/kg, po by LC-MS/MS analysis | Mus musculus | 1 | ALA4118098 | organism-based format | Scientific Literature | |
| 8. | ALA4120247 | A | Tmax in C57BL/6J mouse at 30 mg/kg, po by LC-MS/MS analysis | Mus musculus | 1 | ALA4118098 | organism-based format | Scientific Literature | |
| 9. | ALA4120248 | A | AUC in C57BL/6J mouse at 30 mg/kg, po by LC-MS/MS analysis | Mus musculus | 1 | ALA4118098 | organism-based format | Scientific Literature | |
| 10. | ALA4120678 | B | Inhibition of MAPKAPK2 (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 11. | ALA4120679 | B | Inhibition of AurA (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 12. | ALA4120680 | B | Inhibition of PKC-zeta (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 13. | ALA4120681 | B | Inhibition of RSK1 (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 14. | ALA4120682 | B | Inhibition of PRAK (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 15. | ALA4120683 | B | Inhibition of Erk1 (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 16. | ALA4120684 | B | Inhibition of PKD2 (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 17. | ALA4120685 | B | Inhibition of CK1-delta (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 18. | ALA4120686 | B | Inhibition of CHK1 (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 19. | ALA4120687 | B | Inhibition of ABL (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature | |
| 20. | ALA4120688 | B | Inhibition of FYN (unknown origin) at 0.164 uM relative to control | Homo sapiens | 1 | ALA4118098 | single protein format | Scientific Literature |
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