| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4123721 | Binding | Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assay | Homo sapiens | 15 | ALA4118199 | single protein format | Scientific Literature | |
| 2. | ALA4123722 | Binding | Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate after 60 mins by fluorescence assay | Homo sapiens | 15 | ALA4118199 | single protein format | Scientific Literature | |
| 3. | ALA4123723 | Binding | Selectivity ratio of IC50 for human 20S constitutive proteasome beta-5 to IC50 for human 20S constitutive proteasome beta-2 | Homo sapiens | 15 | ALA4118199 | assay format | Scientific Literature | |
| 4. | ALA4123727 | Physicochemical | Stability in pH 6.5 PBS buffer at 1 mM after 12 hrs by HPLC analysis | 15 | ALA4118199 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA4123728 | Physicochemical | Stability in pH 7.4 PBS buffer at 1 mM after 1 hr by HPLC analysis | 15 | ALA4118199 | small-molecule physicochemical format | Scientific Literature | ||
| 6. | ALA4123729 | Physicochemical | Stability in pH 7.4 PBS buffer at 1 mM after 6 hrs by HPLC analysis | 15 | ALA4118199 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA4123730 | Physicochemical | Stability in pH 8 PBS buffer at 1 mM after 2 hrs by HPLC analysis | 15 | ALA4118199 | small-molecule physicochemical format | Scientific Literature |
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