| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4137466 | B | Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assay | Homo sapiens | 39 | single protein format | Scientific Literature | ||
| 2. | ALA4137467 | B | Inhibition of human DNMT1 using polydeoxyinosine polydeoxycytosine DNA as substrate after 15 mins in presence of SAM by TR-FRET assay | Homo sapiens | 39 | single protein format | Scientific Literature | ||
| 3. | ALA4137469 | F | Growth inhibition of human CEMO1 cells after 48 hrs by MTS assay | Homo sapiens | 13 | assay format | Scientific Literature | ||
| 4. | ALA4137476 | F | Growth inhibition of human OCI-LY3 cells at 1 uM after 48 hrs by MTS assay relative to control | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 5. | ALA4137477 | B | Inhibition of recombinant human GLP using histone H3 peptide as substrate after 120 mins in presence of [3H]SAM by radiometric assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 6. | ALA4137479 | F | Growth inhibition of human OCI-LY10 cells at 1 uM after 48 hrs by MTS assay relative to control | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 7. | ALA4137480 | F | Growth inhibition of human MV4-11 cells after 48 hrs by MTS assay | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 8. | ALA4137481 | A | Growth inhibition of human THLE2 cells after 72 hrs by MTS assay | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 9. | ALA4137482 | B | Competitive inhibition of human G9a using 40 to 2560 nM biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 10. | ALA4137483 | B | Competitive inhibition of human DNMT1 using 1 to 100 ug/ml polydeoxyinosine polydeoxycytosine DNA as substrate after 15 mins in presence of SAM by TR-FRET assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4137484 | B | Non-competitive inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of 2 to 640 uM SAM by TR-FRET assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4137485 | B | Non-competitive inhibition of human DNMT1 using polydeoxyinosine polydeoxycytosine DNA as substrate after 15 mins in presence of 1 to 20 uM SAM by TR-FRET assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4137486 | B | Inhibition of recombinant human N-terminal GST-tagged DNMT3A (1 to 913 residues) expressed in baculovirus infected Sf9 cells at 10 uM relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 14. | ALA4137487 | B | Inhibition of recombinant mouse N-terminal His/C-terminal FLAG-tagged DNMT3B (2 to 859 residues) expressed in baculovirus infected Sf9 cells at 10 uM relative to control | Mus musculus | 2 | cell-based format | Scientific Literature |
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