# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4155089 | B | Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assay | Homo sapiens | 18 | ALA4152267 | assay format | Scientific Literature | |
2. | ALA4155090 | B | Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate after 30 mins by ADP-Glo reagent based luminescence assay | Rattus norvegicus | 6 | ALA4152267 | assay format | Scientific Literature | |
3. | ALA4155091 | B | Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assay | Homo sapiens | 6 | ALA4152267 | protein complex format | Scientific Literature | |
4. | ALA4155092 | B | Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30 mins by ADP-Glo reagent based luminescence assay | Homo sapiens | 6 | ALA4152267 | cell-based format | Scientific Literature | |
5. | ALA4155093 | B | Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as substrate after 30 mins by ADP-Glo reagent based luminescence assay | Homo sapiens | 6 | ALA4152267 | assay format | Scientific Literature | |
6. | ALA4155094 | B | Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based luminescence assay | Mus musculus | 6 | ALA4152267 | assay format | Scientific Literature | |
7. | ALA4155095 | B | Inhibition of porcine brain CK1delta/epsilon using RRKHAAIGSpAYSITA as substrate after 30 mins by ADP-Glo reagent based luminescence assay | Sus scrofa | 6 | ALA4152267 | assay format | Scientific Literature | |
8. | ALA4155096 | B | Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assay | Sus scrofa | 6 | ALA4152267 | assay format | Scientific Literature | |
9. | ALA4155097 | F | Cytotoxicity against human KU812 cells assessed as reduction in cell viability after 48 hrs by MTT assay | Homo sapiens | 6 | ALA4152267 | cell-based format | Scientific Literature |