| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4158156 | Functional | Agonist activity to human FFA2R expressed in HEK293T cells assessed as induction beta-arrestin-2 recruitment after 10 mins by BRET assay | Homo sapiens | 30 | ALA4152367 | cell-based format | Scientific Literature | |
| 2. | ALA4158157 | Functional | Agonist activity to human FFA2R expressed in HEK293T cells assessed as induction beta-arrestin-2 recruitment after 10 mins by BRET assay relative to propionate | Homo sapiens | 27 | ALA4152367 | cell-based format | Scientific Literature | |
| 3. | ALA4158158 | Functional | Agonist activity at human FFA2R expressed in Flp-InT-REx 293 cells assessed as reduction of forskolin-induced cAMP production after 30 mins by TR-FRET assay | Homo sapiens | 25 | ALA4152367 | cell-based format | Scientific Literature | |
| 4. | ALA4158159 | Functional | Agonist activity at human FFA2R expressed in Flp-InT-REx 293 cells assessed as reduction of forskolin-induced cAMP production after 30 mins by TR-FRET assay relative to propionate | Homo sapiens | 25 | ALA4152367 | cell-based format | Scientific Literature | |
| 5. | ALA4158163 | Binding | Displacement of [3H]-GLPG0974 from human FFA2 expressed in Flp-InT-REx 293 cell membranes after 2 hrs by liquid scintillation spectrometry | Homo sapiens | 6 | ALA4152367 | cell-based format | Scientific Literature | |
| 6. | ALA4158164 | Functional | Agonist activity at FFA3R (unknown origin) up to 100 uM | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 7. | ALA4158165 | Functional | Agonist activity at human FFA1R expressed in HEK293 cells assessed as induction of calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | cell-based format | Scientific Literature | |
| 8. | ALA4158166 | Functional | Antagonist activity at human FFA1 receptor expressed in HEK293 cells assessed as inhibition of linoleic acid-induced calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | cell-based format | Scientific Literature | |
| 9. | ALA4158167 | Functional | Agonist activity at human FFA4 receptor expressed in HEK293 cells assessed as induction of calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | cell-based format | Scientific Literature | |
| 10. | ALA4158168 | Functional | Antagonist activity at human FFA4 receptor expressed in HEK293 cells assessed as inhibition of GW9508-induced of calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | cell-based format | Scientific Literature | |
| 11. | ALA4158169 | Binding | Agonist activity at human PPARalpha expressed in Escherichia coli assessed as induction of calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 12. | ALA4158170 | Binding | Antagonist activity at human PPARalpha expressed in Escherichia coli assessed as inhibition of GW9662-induced calcium flux at 10 uM by alpha screen assay | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 13. | ALA4158171 | Binding | Agonist activity at human PPARgamma expressed in Escherichia coli assessed as induction of calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 14. | ALA4158172 | Binding | Antagonist activity at human PPARgamma expressed in Escherichia coli assessed as inhibition of rosiglitazone-induced calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 15. | ALA4158173 | Binding | Agonist activity at human PPARdelta expressed in Escherichia coli assessed as induction of calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 16. | ALA4158174 | Binding | Antagonist activity at human PPARdelta expressed in Escherichia coli assessed as inhibition of GW0742-induced calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 17. | ALA4158175 | Binding | Agonist activity at human LXRalpha expressed in Escherichia coli assessed as induction of calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 18. | ALA4158176 | Binding | Antagonist activity at human LXRalpha expressed in Escherichia coli assessed as inhibition of T0901317-induced calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 19. | ALA4158177 | Binding | Agonist activity at human LXRbeta expressed in Escherichia coli assessed as induction of calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature | |
| 20. | ALA4158178 | Binding | Antagonist activity at human LXRbeta expressed in Escherichia coli assessed as inhibition of T0901317-induced calcium flux at 10 uM by fluorimetry | Homo sapiens | 1 | ALA4152367 | assay format | Scientific Literature |
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