| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4180809 | B | Inhibition of recombinant human N-terminal GST-His6 tagged PDGFRalpha (Q551 to L1089 residues) expressed in Sf9 insect cells using poly(Ala,Glu,Lys,Tyr)6:2:5:1 hydrobromide as substrate in presence of [gamma-33P]ATP | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 2. | ALA4180810 | B | Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-33P]ATP | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 3. | ALA4180811 | F | Cytotoxicity against human HCC827 cells assessed as growth inhibition after 72 hrs by calcein-AM dye based fluorescence assay | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 4. | ALA4180812 | F | Cytotoxicity against human BT474 cells assessed as growth inhibition after 72 hrs by calcein-AM dye based fluorescence assay | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 5. | ALA4180813 | F | Cytotoxicity against human MCF7 cells assessed as growth inhibition after 72 hrs by calcein-AM dye based fluorescence assay | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 6. | ALA4180814 | F | Cytotoxicity against human K562 cells assessed as growth inhibition after 72 hrs by calcein-AM dye based fluorescence assay | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 7. | ALA4180815 | F | Cytotoxicity against human EOL-1 cells assessed as growth inhibition after 72 hrs by calcein-AM dye based fluorescence assay | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 8. | ALA4180816 | F | Cell cycle arrest in human EOL-1 cells assessed as G1/G2-M ratio at GI50 concentration after 24 hrs by propidium iodide staining-based flow cytometry relative to control | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 9. | ALA4180817 | F | Cell cycle arrest in human HCC827 cells assessed as G1/G2-M ratio at GI50 concentration after 24 hrs by propidium iodide staining-based flow cytometry relative to control | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 10. | ALA4180818 | F | Cell cycle arrest in human K562 cells assessed as G1/G2-M ratio at GI50 concentration after 24 hrs by propidium iodide staining-based flow cytometry relative to control | Homo sapiens | 25 | ALA4177643 | cell-based format | Scientific Literature | |
| 11. | ALA4180845 | B | Inhibition of rat liver AMPK assessed as residual activity at 1 uM after 30 mins in presence of [gamma-33P]ATP relative to control relative to control | Rattus norvegicus | 1 | ALA4177643 | assay format | Scientific Literature | |
| 12. | ALA4180846 | B | Inhibition of recombinant human full length His6-tagged Aurora B expressed in Sf21 insect cells assessed as residual activity at 1 uM using LRRLSLGLRRLSLGLRRLSLGLRRLSLG as substrate after 30 mins in presence of [gamma-33P]ATP relative to control | Homo sapiens | 1 | ALA4177643 | cell-based format | Scientific Literature | |
| 13. | ALA4180847 | B | Inhibition of BTK (unknown origin) assessed as residual activity at 1 uM relative to control | Homo sapiens | 1 | ALA4177643 | single protein format | Scientific Literature | |
| 14. | ALA4180848 | B | Inhibition of human full length CAMK1 assessed as residual activity at 1 uM after 30 mins in presence of [gamma-33P]ATP relative to control | Homo sapiens | 1 | ALA4177643 | single protein format | Scientific Literature | |
| 15. | ALA4180849 | B | Inhibition of recombinant human full length GST-tagged CAMKKbeta expressed in Escherichia coli assessed as residual activity at 1 uM using AKPKGNKDYHLQTCCGSLAYRRR as substrate after 30 mins in presence of [gamma-33P]ATP relative to control | Homo sapiens | 1 | ALA4177643 | assay format | Scientific Literature | |
| 16. | ALA4180850 | B | Inhibition of recombinant human full length GST-tagged CK1delta (1 to 294 residues) expressed in Escherichia coli assessed as residual activity at 1 uM after 30 mins in presence of [gamma-33P]ATP relative to control | Homo sapiens | 1 | ALA4177643 | assay format | Scientific Literature | |
| 17. | ALA4180851 | B | Inhibition of human full length CK2 assessed as residual activity at 1 uM after 30 mins in presence of [gamma-33P]ATP relative to control | Homo sapiens | 1 | ALA4177643 | protein format | Scientific Literature | |
| 18. | ALA4180852 | B | Inhibition of recombinant human full length GST-tagged DYRK1A (1 to 499 residues) expressed in Escherichia coli assessed as residual activity at 1 uM using KKISGRLSPIMTEQ as substrate after 30 mins in presence of [gamma-33P]ATP relative to control | Homo sapiens | 1 | ALA4177643 | assay format | Scientific Literature | |
| 19. | ALA4180853 | B | Inhibition of recombinant human full length GST-tagged EF2K expressed in Escherichia coli assessed as residual activity at 1 uM using RKKFGESKTKTKEFL as substrate after 30 mins in presence of [gamma-33P]ATP relative to control | Homo sapiens | 1 | ALA4177643 | assay format | Scientific Literature | |
| 20. | ALA4180854 | B | Inhibition of EPHA2 (unknown origin) assessed as residual activity at 1 uM relative to control | Homo sapiens | 1 | ALA4177643 | single protein format | Scientific Literature |
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