| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4189162 | B | Agonist activity at human N-terminal alphaHis-SUMO-tagged ERRgamma-LBD (229 to 458 residues) expressed in Escherichia coli BL21 gold (DE3) cells assessed as decrease in RIP140 peptide recruitment after 2 hrs by TR-FRET assay | Homo sapiens | 78 | ALA4184311 | cell-based format | Scientific Literature | |
| 2. | ALA4189163 | B | Agonist activity at Gal4 fused ERRgamma-LBD (unknown origin) expressed in HEK293T cells after 20 hrs by UAS-luciferase reporter gene assay | Homo sapiens | 2 | ALA4184311 | cell-based format | Scientific Literature | |
| 3. | ALA4189164 | A | Half life in human liver microsomes at 1 uM in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 6 | ALA4184311 | microsome format | Scientific Literature | |
| 4. | ALA4189165 | A | Half life in mouse liver microsomes at 1 uM in presence of NADPH by LC-MS/MS analysis | Mus musculus | 6 | ALA4184311 | microsome format | Scientific Literature | |
| 5. | ALA4189166 | A | Half life in rat liver microsomes at 1 uM in presence of NADPH by LC-MS/MS analysis | Rattus norvegicus | 6 | ALA4184311 | microsome format | Scientific Literature | |
| 6. | ALA4189169 | B | Agonist activity at alphaHis-SUMO-tagged ERRalpha-LBD (unknown origin) assessed as decrease in RIP140 peptide recruitment by TR-FRET assay | Homo sapiens | 6 | ALA4184311 | single protein format | Scientific Literature | |
| 7. | ALA4189170 | B | Agonist activity at alphaHis-SUMO-tagged ERRbeta-LBD (unknown origin) assessed as decrease in RIP140 peptide recruitment by TR-FRET assay | Homo sapiens | 6 | ALA4184311 | single protein format | Scientific Literature | |
| 8. | ALA4189171 | B | Agonist activity at Herpes simplex virus Gal4 fused VP16-LBD expressed in HEK293T cells after 20 hrs by UAS-luciferase reporter gene assay | unidentified herpesvirus | 2 | ALA4184311 | cell-based format | Scientific Literature | |
| 9. | ALA4189172 | B | Selectivity ratio of EC50 for alphaHis-SUMO-tagged ERRbeta-LBD (unknown origin) to EC50 for human N-terminal alphaHis-SUMO-tagged ERRgamma-LBD (229 to 458 residues) expressed in Escherichia coli BL21 gold (DE3) cells | Homo sapiens | 4 | ALA4184311 | cell-based format | Scientific Literature |
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